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Jagabandhu Das
Bristol-Myers Squibb Research and Development
PO Box 4000
Princeton
NJ 08543-4000
USA
Name/email consistency: high
- Pyrazolo-pyrimidines: a novel heterocyclic scaffold for potent and selective p38 alpha inhibitors. Das, J., Moquin, R.V., Pitt, S., Zhang, R., Shen, D.R., McIntyre, K.W., Gillooly, K., Doweyko, A.M., Sack, J.S., Zhang, H., Kiefer, S.E., Kish, K., McKinnon, M., Barrish, J.C., Dodd, J.H., Schieven, G.L., Leftheris, K. Bioorg. Med. Chem. Lett. (2008)
- Discovery and SAR of 2-amino-5-[(thiomethyl)aryl]thiazoles as potent and selective Itk inhibitors. Das, J., Liu, C., Moquin, R.V., Lin, J., Furch, J.A., Spergel, S.H., Doweyko, A.M., McIntyre, K.W., Shuster, D.J., O'Day, K.D., Penhallow, B., Hung, C.Y., Kanner, S.B., Lin, T.A., Dodd, J.H., Barrish, J.C., Wityak, J. Bioorg. Med. Chem. Lett. (2006)
- Discovery and SAR of 2-amino-5-(thioaryl)thiazoles as potent and selective Itk inhibitors. Das, J., Furch, J.A., Liu, C., Moquin, R.V., Lin, J., Spergel, S.H., McIntyre, K.W., Shuster, D.J., O'Day, K.D., Penhallow, B., Hung, C.Y., Doweyko, A.M., Kamath, A., Zhang, H., Marathe, P., Kanner, S.B., Lin, T.A., Dodd, J.H., Barrish, J.C., Wityak, J. Bioorg. Med. Chem. Lett. (2006)
- 2-aminothiazole as a novel kinase inhibitor template. Structure-activity relationship studies toward the discovery of N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1- piperazinyl)]-2-methyl-4-pyrimidinyl]amino)]-1,3-thiazole-5-carboxamide (dasatinib, BMS-354825) as a potent pan-Src kinase inhibitor. Das, J., Chen, P., Norris, D., Padmanabha, R., Lin, J., Moquin, R.V., Shen, Z., Cook, L.S., Doweyko, A.M., Pitt, S., Pang, S., Shen, D.R., Fang, Q., de Fex, H.F., McIntyre, K.W., Shuster, D.J., Gillooly, K.M., Behnia, K., Schieven, G.L., Wityak, J., Barrish, J.C. J. Med. Chem. (2006)
- Molecular design, synthesis, and structure-Activity relationships leading to the potent and selective p56(lck) inhibitor BMS-243117. Das, J., Lin, J., Moquin, R.V., Shen, Z., Spergel, S.H., Wityak, J., Doweyko, A.M., DeFex, H.F., Fang, Q., Pang, S., Pitt, S., Shen, D.R., Schieven, G.L., Barrish, J.C. Bioorg. Med. Chem. Lett. (2003)
- Discovery of 2-amino-heteroaryl-benzothiazole-6-anilides as potent p56(lck) inhibitors. Das, J., Moquin, R.V., Lin, J., Liu, C., Doweyko, A.M., DeFex, H.F., Fang, Q., Pang, S., Pitt, S., Shen, D.R., Schieven, G.L., Barrish, J.C., Wityak, J. Bioorg. Med. Chem. Lett. (2003)
- Thrombin active site inhibitors: chemical synthesis, in vitro and in vivo pharmacological profile of a novel and selective agent BMS-189090 and analogues. Das, J., Kimball, S.D., Reid, J.A., Wang, T.C., Lau, W.F., Roberts, D.G., Seiler, S.M., Schumacher, W.A., Ogletree, M.L. Bioorg. Med. Chem. Lett. (2002)
- Molecular design and structure--activity relationships leading to the potent, selective, and orally active thrombin active site inhibitor BMS-189664. Das, J., Kimball, S.D., Hall, S.E., Han, W.C., Iwanowicz, E., Lin, J., Moquin, R.V., Reid, J.A., Sack, J.S., Malley, M.F., Chang, C.Y., Chong, S., Wang-Iverson, D.B., Roberts, D.G., Seiler, S.M., Schumacher, W.A., Ogletree, M.L. Bioorg. Med. Chem. Lett. (2002)
