Chemical Compound Review:
Delt-II (4S)-4-[[1-[[(1S)-1- (aminocarbonylmethylca...
Synonyms:
Deltorphin-II, Deltorphin II, Delt II, LS-72217, AC1L3XB1, ...
Benamar,
Rawls,
Geller,
Adler,
Gustafsson,
Afrah,
Stiller,
Di Giannuario,
Pieretti,
Sagratella,
Loizzo,
Salmi,
Kela,
Arvidsson,
Wahlestedt,
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- Antihyperalgesic effects of delta opioid agonists in a rat model of chronic inflammation. Fraser, G.L., Gaudreau, G.A., Clarke, P.B., Ménard, D.P., Perkins, M.N. Br. J. Pharmacol. (2000)
- Functional interactions between delta- and mu-opioid receptors in rat thermoregulation. Salmi, P., Kela, J., Arvidsson, U., Wahlestedt, C. Eur. J. Pharmacol. (2003)
- Effects of mu, kappa or delta opioids administered by pellet or pump on oral Salmonella infection and gastrointestinal transit. Feng, P., Rahim, R.T., Cowan, A., Liu-Chen, L.Y., Peng, X., Gaughan, J., Meissler, J.J., Adler, M.W., Eisenstein, T.K. Eur. J. Pharmacol. (2006)
- The role of delta-opioid receptor subtypes in neuropathic pain. Mika, J., Przewłocki, R., Przewłocka, B. Eur. J. Pharmacol. (2001)
- The effects of delta agonists on locomotor activity in habituated and non-habituated rats. Fraser, G.L., Parenteau, H., Tu, T.M., Ducharme, J., Perkins, M.N., Clarke, P.B. Life Sci. (2000)
- Activity of the delta-opioid receptor is partially reduced, whereas activity of the kappa-receptor is maintained in mice lacking the mu-receptor. Matthes, H.W., Smadja, C., Valverde, O., Vonesch, J.L., Foutz, A.S., Boudinot, E., Denavit-Saubié, M., Severini, C., Negri, L., Roques, B.P., Maldonado, R., Kieffer, B.L. J. Neurosci. (1998)
- The alpha2a adrenergic receptor subtype mediates spinal analgesia evoked by alpha2 agonists and is necessary for spinal adrenergic-opioid synergy. Stone, L.S., MacMillan, L.B., Kitto, K.F., Limbird, L.E., Wilcox, G.L. J. Neurosci. (1997)
- Deltorphin II-induced rapid desensitization of delta-opioid receptor requires both phosphorylation and internalization of the receptor. Law, P.Y., Kouhen, O.M., Solberg, J., Wang, W., Erickson, L.J., Loh, H.H. J. Biol. Chem. (2000)
- DPDPE-UK14,304 synergy is retained in mu opioid receptor knockout mice. Guo, X.H., Fairbanks, C.A., Stone, L.S., Loh, H.H. Pain (2003)
- The distribution of the anti-HIV drug, 2'3'-dideoxycytidine (ddC), across the blood-brain and blood-cerebrospinal fluid barriers and the influence of organic anion transport inhibitors. Gibbs, J.E., Thomas, S.A. J. Neurochem. (2002)
- Dexamethasone modulates hypotension induced by opioids in anaesthetised rats. Sorrentino, R., Capasso, A., d'Emmanuele di Villa Bianca, R., Pinto, A. Eur. J. Pharmacol. (2001)
- Intrahypothalamic injection of deltorphin-II alters body temperature in rats. Benamar, K., Rawls, S.M., Geller, E.B., Adler, M.W. Brain Res. (2004)
- Interactions between angiotensin II and delta opioid receptor subtype agonists upon water intake in rats. Yu, W.Z., Bodnar, R.J. Peptides (1997)
- Characterization of [3H]naltrindole binding to delta opioid receptors in rat brain. Yamamura, M.S., Horvath, R., Toth, G., Otvos, F., Malatynska, E., Knapp, R.J., Porreca, F., Hruby, V.J., Yamamura, H.I. Life Sci. (1992)
- The role of backbone conformation in deltorphin II binding: a QSAR study of new analogues modified in the 5-, 6-positions of the address domain. Schullery, S.E., Rodgers, D.W., Tripathy, S., Jayamaha, D.E., Sanvordekar, M.D., Renganathan, K., Mousigian, C., Heyl, D.L. Bioorg. Med. Chem. (2001)
- Comparison between delta-opioid receptor functional response and autoradiographic labeling in rat brain and spinal cord. Pradhan, A.A., Clarke, P.B. J. Comp. Neurol. (2005)
- Lack of dependence and rewarding effects of deltorphin II in mu-opioid receptor-deficient mice. Hutcheson, D.M., Matthes, H.W., Valjent, E., Sánchez-Blázquez, P., Rodríguez-Díaz, M., Garzón, J., Kieffer, B.L., Maldonado, R. Eur. J. Neurosci. (2001)
- Organic anion-transporting polypeptides mediate transport of opioid peptides across blood-brain barrier. Gao, B., Hagenbuch, B., Kullak-Ublick, G.A., Benke, D., Aguzzi, A., Meier, P.J. J. Pharmacol. Exp. Ther. (2000)
- Moxonidine, a selective imidazoline/alpha(2) adrenergic receptor agonist, synergizes with morphine and deltorphin II to inhibit substance P-induced behavior in mice. Fairbanks, C.A., Posthumus, I.J., Kitto, K.F., Stone, L.S., Wilcox, G.L. Pain (2000)
- The delta agonists DPDPE and deltorphin II recruit predominantly mu receptors to produce thermal analgesia: a parallel study of mu, delta and combinatorial opioid receptor knockout mice. Scherrer, G., Befort, K., Contet, C., Becker, J., Matifas, A., Kieffer, B.L. Eur. J. Neurosci. (2004)
- Functional characterization of opioid receptor ligands by aequorin luminescence-based calcium assay. Fichna, J., Gach, K., Piestrzeniewicz, M., Burgeon, E., Poels, J., Broeck, J.V., Janecka, A. J. Pharmacol. Exp. Ther. (2006)
- dextro- and levo-morphine attenuate opioid delta and kappa receptor agonist produced analgesia in mu-opioid receptor knockout mice. Wu, H.E., Sun, H.S., Terashivili, M., Schwasinger, E., Sora, I., Scott Hall, F., Uhl, G.R., Tseng, L.F. Eur. J. Pharmacol. (2006)
- Deltorphin II enhances extracellular levels of dopamine in the nucleus accumbens via opioid receptor-independent mechanisms. Murakawa, K., Hirose, N., Takada, K., Suzuki, T., Nagase, H., Cools, A.R., Koshikawa, N. Eur. J. Pharmacol. (2004)
- Respiratory function in adult mice lacking the mu-opioid receptor: role of delta-receptors. Morin-Surun, M.P., Boudinot, E., Dubois, C., Matthes, H.W., Kieffer, B.L., Denavit-Saubié, M., Champagnat, J., Foutz, A.S. Eur. J. Neurosci. (2001)
- [L-Ala3]DPDPE: a new enkephalin analog with a unique opioid receptor activity profile. Further evidence of delta-opioid receptor multiplicity. Haaseth, R.C., Horan, P.J., Bilsky, E.J., Davis, P., Zalewska, T., Slaninova, J., Yamamura, H.I., Weber, S.J., Davis, T.P., Porreca, F. J. Med. Chem. (1994)
- delta-opioid receptor mobilization of intracellular calcium in SH-SY5Y cells: lack of evidence for delta-receptor subtypes. Connor, M.A., Keir, M.J., Henderson, G. Neuropharmacology (1997)
- Morphine-induced in vivo release of spinal cholecystokinin is mediated by delta-opioid receptors--effect of peripheral axotomy. Gustafsson, H., Afrah, A.W., Stiller, C.O. J. Neurochem. (2001)
- Repeated {delta}1-opioid receptor stimulation reduces {delta}2-opioid receptor responses in the SA node. Deo, S.H., Johnson-Davis, S., Barlow, M.A., Yoshishige, D., Caffrey, J.L. Am. J. Physiol. Heart Circ. Physiol. (2006)
- Dexamethasone blocking effects on mu- and delta-opioid-induced seizures involves kappa-opioid activity in the rabbit. Di Giannuario, A., Pieretti, S., Sagratella, S., Loizzo, A. Neuropsychobiology (2001)
- Binding of agonists, antagonists and inverse agonists to the human delta-opioid receptor produces distinctly different conformational states distinguishable by plasmon-waveguide resonance spectroscopy. Salamon, Z., Hruby, V.J., Tollin, G., Cowell, S. J. Pept. Res. (2002)