Giampaolo Primofiore
Dipartimento di Scienze Farmaceutiche
Università di Pisa
Via Bonanno 6
56126 Pisa
Italy
Name/email consistency: high
- Novel N-substituted indol-3-ylglyoxylamides probing the LDi and L1/L2 lipophilic regions of the benzodiazepine receptor site in search for subtype-selective ligands. Primofiore, G., Taliani, S., Da Settimo, F., Marini, A.M., La Motta, C., Simorini, F., Patrizi, M.P., Sergianni, V., Novellino, E., Greco, G., Cosimelli, B., Calderone, V., Montali, M., Besnard, F., Martini, C. J. Med. Chem. (2007)
- Synthesis and benzodiazepine receptor affinity of derivatives of the new tricyclic heteroaromatic system pyrido[3',2':5,6]thiopyrano[4,3-c]pyridazin-3(2H,5H)-one. Primofiore, G., Da Settimo, F., Marini, A.M., Simorini, F., La Motta, C., Taliani, S., Laneri, S., Trincavelli, L., Martini, C. Arch. Pharm. (Weinheim) (2005)
- High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives. Primofiore, G., Da Settimo, F., Taliani, S., Salerno, S., Novellino, E., Greco, G., Cosimelli, B., Besnard, F., Costa, B., Montali, M., Martini, C. J. Med. Chem. (2005)
- Geometrically constrained analogues of N-benzylindolylglyoxylylamides: [1, 2, 4]triazino[4, 3-a]benzimidazol-4(10H)-one derivatives as potential new ligands at the benzodiazepine receptor. Primofiore, G., Da Settimo, F., Taliani, S., Marini, A.M., Simorini, F., Novellino, E., Greco, G., Trincavelli, L., Martini, C. Arch. Pharm. (Weinheim) (2003)
- Novel N-(arylalkyl)indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships. Primofiore, G., Settimo, F.D., Taliani, S., Marini, A.M., Novellino, E., Greco, G., Lavecchia, A., Besnard, F., Trincavelli, L., Costa, B., Martini, C. J. Med. Chem. (2001)









