Chemical Compound Review:
Pacinone 9-chloro-6-phenyl-2-(2,2,2- trifluoroethyl)...
Synonyms:
Halazepam, Paxipam, Halazepamum, CHEMBL970, Paxipam (TN), ...
- Selective affinity of 1-N-trifluoroethyl benzodiazepines for cerebellar type 1 receptor sites. Iorio, L.C., Barnett, A., Billard, W. Life Sci. (1984)
- Effectiveness of bedtime dosing of benzodiazepines: a placebo-controlled comparison of halazepam and clorazepate. Aden, G.C., O'Hair, D.E. Clinical therapeutics. (1980)
- Multiple-dose halazepam kinetics. Chung, M., Hilbert, J.M., Gural, R.P., Radwanski, E., Symchowicz, S., Zampaglione, N. Clin. Pharmacol. Ther. (1984)
- Clinical pharmacokinetics of the newer benzodiazepines. Greenblatt, D.J., Divoll, M., Abernethy, D.R., Ochs, H.R., Shader, R.I. Clinical pharmacokinetics. (1983)
- Liquid chromatographic assay and pharmacokinetics of halazepam and its metabolite in humans. Gupta, S.K., Ellinwood, E.H. Journal of pharmaceutical sciences. (1990)
- Metabolism of halazepam by rat liver microsomes: stereoselective formation and N-dealkylation of 3-hydroxyhalazepam. Lu, X.L., Yang, S.K. Chirality. (1990)
- Pharmacology, efficacy, and adverse effects of halazepam, a new benzodiazepine. Fann, W.E., Pitts, W.M., Wheless, J.C. Pharmacotherapy (1982)
- Autoradiographic demonstration of the selectivity of two 1-N-trifluoroethyl benzodiazepines for the BZD-1 receptors in the rat brain. Wamsley, J.K., Golden, J.S., Yamamura, H.I., Barnett, A. Pharmacol. Biochem. Behav. (1985)
- Diazepam and halazepam in anxiety: some prognostic indicators. Rickels, K., Case, W.G., Chung, H., Downing, R.W., Vlahovich, J. International pharmacopsychiatry. (1978)
- The effects of one-day treatment of anxiety with high doses of halazepam. Kellner, R., Bruzzese, D., Winslow, W.W., Rada, R.T., Wall, F.J. Journal of clinical pharmacology. (1978)