Yoshiaki Shimada
Institute for Drug Discovery Research
Yamanouchi Pharmaceultical Co
Ltd, Tsukuba-shi
Ibaraki
Japan
Name/email consistency: high
- Stereoselective synthesis of methyl (Z)-(4,4-difluoro-2,3,4,5-tetrahydro-1H-1-benzazepin-5-ylidene)acetate using a dianion Horner-Wadsworth-Emmons reagent. Shimada, Y., Akane, H., Taniguchi, N., Matsuhisa, A., Kawano, N., Tanaka, A. Chem. Pharm. Bull. (2005)
- Preparation of highly potent and selective non-peptide antagonists of the arginine vasopressin V1A receptor by introduction of a 2-ethyl-1H-1-imidazolyl group. Shimada, Y., Akane, H., Taniguchi, N., Matsuhisa, A., Kawano, N., Kikuchi, K., Yatsu, T., Tahara, A., Tomura, Y., Kusayama, T., Wada, K., Tsukada, J., Tsunoda, T., Tanaka, A. Chem. Pharm. Bull. (2005)
- Preparation of non-peptide, highly potent and selective antagonists of arginine vasopressin V1A receptor by introduction of alkoxy groups. Shimada, Y., Taniguchi, N., Matsuhisa, A., Yatsu, T., Tahara, A., Tanaka, A. Chem. Pharm. Bull. (2003)
- Highly potent and orally active non-peptide arginine vasopressin antagonists for both V1A and V2 receptors: synthesis and pharmacological properties of 4'-[(4,4-difluoro-5-methylidene-2,3,4,5-tetrahydro-1H-1-benzoazepin-1-y l)carbonyl]-2-phenylbenzanilide derivatives. Shimada, Y., Taniguchi, N., Matsuhisa, A., Sakamoto, K., Yatsu, T., Tanaka, A. Chem. Pharm. Bull. (2000)
