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Dharmarajan Sriram

Medicinal Chemistry & Antimycobacterial Research Laboratory

Pharmacy Group

Birla Institute of Technology & Science - Pilani

Hyderabad Campus

India

[email]@bits-pilani.ac.in

Name/email consistency: high

 
 
 
 
 
 
 

Affiliation

  • Medicinal Chemistry & Antimycobacterial Research Laboratory, Pharmacy Group, Birla Institute of Technology & Science - Pilani, Hyderabad Campus, India. 2003 - 2010

References

  1. Synthesis and antimycobacterial evaluation of novel Phthalazin-4-ylacetamides against log- and starved phase cultures. Sriram, D., Yogeeswari, P., Senthilkumar, P., Sangaraju, D., Nelli, R., Banerjee, D., Bhat, P., Manjashetty, T.H. Chem. Biol. Drug. Des (2010) [Pubmed]
  2. Efavirenz Mannich bases: synthesis, anti-HIV and antitubercular activities. Sriram, D., Banerjee, D., Yogeeswari, P. J. Enzyme. Inhib. Med. Chem (2009) [Pubmed]
  3. N-Hydroxythiosemicarbazones: synthesis and in vitro antitubercular activity. Sriram, D., Yogeeswari, P., Dhakla, P., Senthilkumar, P., Banerjee, D. Bioorg. Med. Chem. Lett. (2007) [Pubmed]
  4. Antimycobacterial activities of novel 1-(cyclopropyl/tert-butyl/4-fluorophenyl)-1,4-dihydro- 6-nitro-4-oxo-7-(substituted secondary amino)-1,8-naphthyridine-3-carboxylic acid. Sriram, D., Senthilkumar, P., Dinakaran, M., Yogeeswari, P., China, A., Nagaraja, V. J. Med. Chem. (2007) [Pubmed]
  5. Antimycobacterial activity of novel 1-(5-cyclobutyl-1,3-oxazol-2-yl)-3-(sub)phenyl/pyridylthiourea compounds endowed with high activity toward multidrug-resistant Mycobacterium tuberculosis. Sriram, D., Yogeeswari, P., Dinakaran, M., Thirumurugan, R. J. Antimicrob. Chemother. (2007) [Pubmed]
  6. Synthesis and in vitro anti-HIV activities of didanosine prodrugs. Sriram, D., Yogeeswari, P., Babu, N.R., Kurre, P.N. J. Enzyme. Inhib. Med. Chem (2007) [Pubmed]
  7. Synthesis and anti-HIV activity of nevirapine prodrugs. Sriram, D., Yogeeswari, P., Kishore, M.R. Pharmazie (2006) [Pubmed]
  8. Synthesis and in vitro antitubercular activity of some 1-[(4-sub)phenyl]-3-(4-{1-[(pyridine-4-carbonyl)hydrazono]ethyl}phenyl)thiourea. Sriram, D., Yogeeswari, P., Madhu, K. Bioorg. Med. Chem. Lett. (2006) [Pubmed]
  9. Synthesis, in vitro and in vivo antimycobacterial activities of diclofenac acid hydrazones and amides. Sriram, D., Yogeeswari, P., Devakaram, R.V. Bioorg. Med. Chem. (2006) [Pubmed]
  10. Abacavir prodrugs: microwave-assisted synthesis and their evaluation of anti-HIV activities. Sriram, D., Yogeeswari, P., Myneedu, N.S., Saraswat, V. Bioorg. Med. Chem. Lett. (2006) [Pubmed]
  11. Synthesis of pyrazinamide Mannich bases and its antitubercular properties. Sriram, D., Yogeeswari, P., Reddy, S.P. Bioorg. Med. Chem. Lett. (2006) [Pubmed]
  12. Gatifloxacin derivatives: synthesis, antimycobacterial activities, and inhibition of Mycobacterium tuberculosis DNA gyrase. Sriram, D., Aubry, A., Yogeeswari, P., Fisher, L.M. Bioorg. Med. Chem. Lett. (2006) [Pubmed]
  13. Synthesis, anti-HIV and antitubercular activities of isatin derivatives. Sriram, D., Yogeeswari, P., Meena, K. Pharmazie (2006) [Pubmed]
  14. Discovery of new antitubercular oxazolyl thiosemicarbazones. Sriram, D., Yogeeswari, P., Thirumurugan, R., Pavana, R.K. J. Med. Chem. (2006) [Pubmed]
  15. Newer aminopyrimidinimino isatin analogues as non-nucleoside HIV-1 reverse transcriptase inhibitors for HIV and other opportunistic infections of AIDS: design, synthesis and biological evaluation. Sriram, D., Bal, T.R., Yogeeswari, P. Farmaco (2005) [Pubmed]
  16. Camptothecin and its analogues: a review on their chemotherapeutic potential. Sriram, D., Yogeeswari, P., Thirumurugan, R., Bal, T.R. Nat. Prod. Res. (2005) [Pubmed]
  17. Synthesis and antimycobacterial evaluation of various 7-substituted ciprofloxacin derivatives. Sriram, D., Yogeeswari, P., Basha, J.S., Radha, D.R., Nagaraja, V. Bioorg. Med. Chem. (2005) [Pubmed]
  18. Combinatorial synthesis of anti-HIV agents--a review. Sriram, D., Yogeeswari, P., Nagappa, A.N. Comb. Chem. High Throughput Screen. (2005) [Pubmed]
  19. Synthesis and in vitro and in vivo antimycobacterial activity of isonicotinoyl hydrazones. Sriram, D., Yogeeswari, P., Madhu, K. Bioorg. Med. Chem. Lett. (2005) [Pubmed]
  20. Synthesis, anti-HIV and antitubercular activities of lamivudine prodrugs. Sriram, D., Yogeeswari, P., Gopal, G. Eur. J. Med. Chem (2005) [Pubmed]
  21. Nevirapine derivatives with broad-spectrum chemotherapeutic properties for the effective treatment of HIV/AIDS. Sriram, D., Srichakravarthy, N., Bal, T.R., Yogeeswari, P. Biomed. Pharmacother. (2005) [Pubmed]
  22. Synthesis of zidovudine prodrugs with broad-spectrum chemotherapeutic properties for the effective treatment of HIV/AIDS. Sriram, D., Srichakravarthy, N., Bal, T.R., Yogeeswari, P. Biomed. Pharmacother. (2005) [Pubmed]
  23. Microwave-assisted synthesis and anti-YFV activity of 2,3-diaryl-1,3-thiazolidin-4-ones. Sriram, D., Yogeeswari, P., Kumar, T.G. J. Pharm. Pharm. Sci (2005) [Pubmed]
  24. Aminopyrimidinimino isatin analogues: design of novel non- nucleoside HIV-1 reverse transcriptase inhibitors with broad-spectrum chemotherapeutic properties. Sriram, D., Bal, T.R., Yogeeswari, P. J. Pharm. Pharm. Sci (2005) [Pubmed]
  25. Aminopyrimidinimino isatin analogues: design and synthesis of novel non- nucleoside HIV-1 reverse transcriptase inhibitors with broad-spectrum anti-microbial properties. Sriram, D., Bal, T.R., Yogeeswari, P. Medicinal. Chemistry. (shāriqah. (united. Arab. Emirates)) (2005) [Pubmed]
  26. Synthesis of stavudine amino acid ester prodrugs with broad-spectrum chemotherapeutic properties for the effective treatment of HIV/AIDS. Sriram, D., Yogeeswari, P., Srichakravarthy, N., Bal, T.R. Bioorg. Med. Chem. Lett. (2004) [Pubmed]
  27. Antituberculous activity of some aryl semicarbazone derivatives. Sriram, D., Yogeeswari, P., Thirumurugan, R. Bioorg. Med. Chem. Lett. (2004) [Pubmed]
  28. Design, synthesis and biological evaluation of novel non-nucleoside HIV-1 reverse transcriptase inhibitors with broad-spectrum chemotherapeutic properties. Sriram, D., Bal, T.R., Yogeeswari, P. Bioorg. Med. Chem. (2004) [Pubmed]
  29. Towards the design and development of agents with broad spectrum chemotherapeutic properties for the effective treatment of HIV / AIDS. Sriram, D., Yogeeswari, P. Curr. Med. Chem. (2003) [Pubmed]
 
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