Gene M. Dubowchik
Bristol-Myers Squibb Pharmaceutical Research Institute
Wallingford
CT 06492-7660
USA
Name/email consistency: high
- An efficient sequence for the preparation of small secondary amine hydrochloride salts for focused library generation without need for distillation or chromatographic purification. Dubowchik, G.M., Michne, J.A., Zuev, D. Bioorg. Med. Chem. Lett. (2004)
- Doxorubicin immunoconjugates containing bivalent, lysosomally-cleavable dipeptide linkages. Dubowchik, G.M., Radia, S., Mastalerz, H., Walker, M.A., Firestone, R.A., Dalton King, H., Hofstead, S.J., Willner, D., Lasch, S.J., Trail, P.A. Bioorg. Med. Chem. Lett. (2002)
- Cathepsin B-labile dipeptide linkers for lysosomal release of doxorubicin from internalizing immunoconjugates: model studies of enzymatic drug release and antigen-specific in vitro anticancer activity. Dubowchik, G.M., Firestone, R.A., Padilla, L., Willner, D., Hofstead, S.J., Mosure, K., Knipe, J.O., Lasch, S.J., Trail, P.A. Bioconjug. Chem. (2002)
- 2-Aryl-2,2-difluoroacetamide FKBP12 ligands: synthesis and X-ray structural studies. Dubowchik, G.M., Vrudhula, V.M., Dasgupta, B., Ditta, J., Chen, T., Sheriff, S., Sipman, K., Witmer, M., Tredup, J., Vyas, D.M., Verdoorn, T.A., Bollini, S., Vinitsky, A. Org. Lett. (2001)
- Fluoresceinated FKBP12 ligands for a high-throughput fluorescence polarization assay. Dubowchik, G.M., Ditta, J.L., Herbst, J.J., Bollini, S., Vinitsky, A. Bioorg. Med. Chem. Lett. (2000)
