Jan Jakubík
Institute of Physiology Academy of Sciences of the Czech Republic
Prague
Czech Republic
Name/email consistency: high
- Negative cooperativity in binding of muscarinic receptor agonists and GDP as a measure of agonist efficacy. Jakubík, J., Janíčková, H., El-Fakahany, E.E., Doležal, V. Br. J. Pharmacol. (2011)
- Divergence of allosteric effects of rapacuronium on binding and function of muscarinic receptors. Jakubík, J., Randáková, A., El-Fakahany, E.E., Dolezal, V. BMC Pharmacol. (2009)
- Determinants of positive cooperativity between strychnine-like allosteric modulators and N-methylscopolamine at muscarinic receptors. Jakubík, J., Dolezal, V. J. Mol. Neurosci. (2006)
- Differences in kinetics of xanomeline binding and selectivity of activation of G proteins at M(1) and M(2) muscarinic acetylcholine receptors. Jakubík, J., El-Fakahany, E.E., Dolezal, V. Mol. Pharmacol. (2006)
- Asparagine, valine, and threonine in the third extracellular loop of muscarinic receptor have essential roles in the positive cooperativity of strychnine-like allosteric modulators. Jakubík, J., Krejcí, A., Dolezal, V. J. Pharmacol. Exp. Ther. (2005)
