Hiroyuki Koshio
Institute for Drug Discovery Research
Yamanouchi Pharmaceutical Co.
Ltd, 21 Miyukigaoka
Tsukuba
Japan
Name/email consistency: high
- Synthesis and biological activity of novel 1,2-disubstituted benzene derivatives as factor Xa inhibitors. Koshio, H., Hirayama, F., Ishihara, T., Shiraki, R., Shigenaga, T., Taniuchi, Y., Sato, K., Moritani, Y., Iwatsuki, Y., Kaku, S., Katayama, N., Kawasaki, T., Matsumoto, Y., Sakamoto, S., Tsukamoto, S. Bioorg. Med. Chem. (2005)
- An easy access to 7-methyl-2-naphthalenecarbonitrile. Koshio, H., Ishihara, T., Yamada, H., Hirayama, F., Matsumoto, Y., Yanagisawa, I. Chem. Pharm. Bull. (2005)
- Synthesis and biological activity of novel 1,4-diazepane derivatives as factor Xa inhibitor with potent anticoagulant and antithrombotic activity. Koshio, H., Hirayama, F., Ishihara, T., Taniuchi, Y., Sato, K., Sakai-Moritani, Y., Kaku, S., Kawasaki, T., Matsumoto, Y., Sakamoto, S., Tsukamoto, S. Bioorg. Med. Chem. (2004)
- Orally active factor Xa inhibitor: synthesis and biological activity of masked amidines as prodrugs of novel 1,4-diazepane derivatives. Koshio, H., Hirayama, F., Ishihara, T., Kaizawa, H., Shigenaga, T., Taniuchi, Y., Sato, K., Moritani, Y., Iwatsuki, Y., Uemura, T., Kaku, S., Kawasaki, T., Matsumoto, Y., Sakamoto, S., Tsukamoto, S. Bioorg. Med. Chem. (2004)