Andrew J. Souers
Metabolic Disease Research
Abbott Laboratories
100 Abbott Park Road
Abbott Park
USA
Name/email consistency: high
- Constrained 7-fluorocarboxychromone-4-aminopiperidine based Melanin-concentrating hormone receptor 1 antagonists: the effects of chirality on substituted indan-1-ylamines. Souers, A.J., Iyengar, R.R., Judd, A.S., Beno, D.W., Gao, J., Zhao, G., Brune, M.E., Napier, J.J., Mulhern, M.M., Lynch, J.K., Freeman, J.C., Wodka, D., Chen, C.J., Falls, H.D., Brodjian, S., Dayton, B.D., Diaz, G.J., Bush, E.N., Shapiro, R., Droz, B.A., Knourek-Segel, V., Hernandez, L.E., Marsh, K.C., Reilly, R.M., Sham, H.L., Collins, C.A., Kym, P.R. Bioorg. Med. Chem. Lett. (2007)
- Identification of 2-(4-benzyloxyphenyl)-N- [1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]acetamide, an orally efficacious melanin-concentrating hormone receptor 1 antagonist for the treatment of obesity. Souers, A.J., Gao, J., Brune, M., Bush, E., Wodka, D., Vasudevan, A., Judd, A.S., Mulhern, M., Brodjian, S., Dayton, B., Shapiro, R., Hernandez, L.E., Marsh, K.C., Sham, H.L., Collins, C.A., Kym, P.R. J. Med. Chem. (2005)
- Synthesis and evaluation of urea-based indazoles as melanin-concentrating hormone receptor 1 antagonists for the treatment of obesity. Souers, A.J., Gao, J., Wodka, D., Judd, A.S., Mulhern, M.M., Napier, J.J., Brune, M.E., Bush, E.N., Brodjian, S.J., Dayton, B.D., Shapiro, R., Hernandez, L.E., Marsh, K.C., Sham, H.L., Collins, C.A., Kym, P.R. Bioorg. Med. Chem. Lett. (2005)
- Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 1. Souers, A.J., Wodka, D., Gao, J., Lewis, J.C., Vasudevan, A., Gentles, R., Brodjian, S., Dayton, B., Ogiela, C.A., Fry, D., Hernandez, L.E., Marsh, K.C., Collins, C.A., Kym, P.R. Bioorg. Med. Chem. Lett. (2004)
- Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 3. Souers, A.J., Wodka, D., Gao, J., Lewis, J.C., Vasudevan, A., Brodjian, S., Dayton, B., Ogiela, C.A., Fry, D., Hernandez, L.E., Marsh, K.C., Collins, C.A., Kym, P.R. Bioorg. Med. Chem. Lett. (2004)