James A. Monn
Core Technology Division
Eli Lilly and Company
Indianapolis
Indiana 46285
USA
Name/email consistency: high
- Synthesis and metabotropic glutamate receptor activity of S-oxidized variants of (-)-4-amino-2-thiabicyclo-[3.1.0]hexane-4,6-dicarboxylate: identification of potent, selective, and orally bioavailable agonists for mGlu2/3 receptors. Monn, J.A., Massey, S.M., Valli, M.J., Henry, S.S., Stephenson, G.A., Bures, M., Hérin, M., Catlow, J., Giera, D., Wright, R.A., Johnson, B.G., Andis, S.L., Kingston, A., Schoepp, D.D. J. Med. Chem. (2007)
- Design, synthesis, and pharmacological characterization of (+)-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (LY354740): a potent, selective, and orally active group 2 metabotropic glutamate receptor agonist possessing anticonvulsant and anxiolytic properties. Monn, J.A., Valli, M.J., Massey, S.M., Wright, R.A., Salhoff, C.R., Johnson, B.G., Howe, T., Alt, C.A., Rhodes, G.A., Robey, R.L., Griffey, K.R., Tizzano, J.P., Kallman, M.J., Helton, D.R., Schoepp, D.D. J. Med. Chem. (1997)
- Synthesis of the four isomers of 4-aminopyrrolidine-2,4-dicarboxylate: identification of a potent, highly selective, and systemically-active agonist for metabotropic glutamate receptors negatively coupled to adenylate cyclase. Monn, J.A., Valli, M.J., Johnson, B.G., Salhoff, C.R., Wright, R.A., Howe, T., Bond, A., Lodge, D., Spangle, L.A., Paschal, J.W., Campbell, J.B., Griffey, K., Tizzano, J.P., Schoepp, D.D. J. Med. Chem. (1996)
