R. Scott Obach
Pharmacokinetics
Pharmacodynamics
and Drug Metabolism
Groton Laboratories
USA
Name/email consistency: high
- Sertraline is metabolized by multiple cytochrome P450 enzymes, monoamine oxidases, and glucuronyl transferases in human: an in vitro study. Obach, R.S., Cox, L.M., Tremaine, L.M. Drug Metab. Dispos. (2005)
- Potent inhibition of human liver aldehyde oxidase by raloxifene. Obach, R.S. Drug Metab. Dispos. (2004)
- Measurement of Michaelis constants for cytochrome P450-mediated biotransformation reactions using a substrate depletion approach. Obach, R.S., Reed-Hagen, A.E. Drug Metab. Dispos. (2002)
- Mechanism of cytochrome P4503A4- and 2D6-catalyzed dehydrogenation of ezlopitant as probed with isotope effects using five deuterated analogs. Obach, R.S. Drug Metab. Dispos. (2001)