Rosario Pignatello
Dipartimento di Scienze del Farmaco
Università degli Studi di Catania
Città Universitaria
viale A. Doria
Italy
Name/email consistency: high
- Amphiphilic erythromycin-lipoamino Acid ion pairs: characterization and in vitro microbiological evaluation. Pignatello, R., Mangiafico, A., Ruozi, B., Puglisi, G., Furneri, P.M. AAPS. PharmSciTech (2011)
- Amphiphilic ion pairs of tobramycin with lipoamino acids. Pignatello, R., Mangiafico, A., Basile, L., Ruozi, B., Furneri, P.M. Eur. J. Med. Chem (2011)
- Effects of liposomal encapsulation on the antioxidant activity of lipophilic prodrugs of idebenone. Pignatello, R., Acquaviva, R., Campisi, A., Raciti, G., Musumeci, T., Puglisi, G. J. Liposome. Res (2011)
- A novel biomaterial for osteotropic drug nanocarriers: synthesis and biocompatibility evaluation of a PLGA-ALE conjugate. Pignatello, R., Cenni, E., Micieli, D., Fotia, C., Salerno, M., Granchi, D., Avnet, S., Sarpietro, M.G., Castelli, F., Baldini, N. Nanomedicine. (Lond) (2009)
- Lipoamino acid prodrugs of paclitaxel: synthesis and cytotoxicity evaluation on human anaplastic thyroid carcinoma cells. Pignatello, R., Paolino, D., Pantò, V., Pistară, V., Calvagno, M.G., Russo, D., Puglisi, G., Fresta, M. Curr. Cancer. Drug. Targets (2009)
- Chitosan glutamate hydrogels with local anesthetic activity for buccal application. Pignatello, R., Basile, L., Puglisi, G. Drug. Deliv (2009)
- Poly(3-hydroxybutyrate-co-epsilon-caprolactone) copolymers and poly(3-hydroxybutyrate-co-3-hydroxyvalerate-co-epsilon-caprolactone) terpolymers as novel materials for colloidal drug delivery systems. Pignatello, R., Musumeci, T., Impallomeni, G., Carnemolla, G.M., Puglisi, G., Ballistreri, A. Eur. J. Pharm. Sci (2009)
- Flurbiprofen derivatives in Alzheimer's disease: synthesis, pharmacokinetic and biological assessment of lipoamino acid prodrugs. Pignatello, R., Pantò, V., Salmaso, S., Bersani, S., Pistarà, V., Kepe, V., Barrio, J.R., Puglisi, G. Bioconjug. Chem. (2008)
- Evaluation of cell tolerability of a series of lipoamino acids using biological membranes and a biomembrane model. Pignatello, R., Noce, C., Campisi, A., Acquaviva, R., Bucolo, C., Puglisi, G., Toth, I. Curr. Drug. Deliv (2007)
- Dexamethasone sodium phosphate-loaded Chitosan based delivery systems for buccal application. Pignatello, R., Stancampiano, A.H., Ventura, C.A., Puglisi, G. J. Drug. Target (2007)
- Conjugation of thymopentin (TP5) with lipoamino acid residues increases the hydrolytic stability and preserves the biological activity. Pignatello, R., Pecora, T.M. Pharmazie (2007)
- Enhancement of drug affinity for cell membranes by conjugation with lipoamino acids II. Experimental and computational evidence using biomembrane models. Pignatello, R., Guccione, S., Castelli, F., Sarpietro, M.G., Giurato, L., Lombardo, M., Puglisi, G., Toth, I. Int. J. Pharm (2006)
- A calorimetric evaluation of the interaction of amphiphilic prodrugs of idebenone with a biomembrane model. Pignatello, R., Intravaia, V.D., Puglisi, G. J. Colloid. Interface. Sci (2006)
- Preparation and characterization of eudragit retard nanosuspensions for the ocular delivery of cloricromene. Pignatello, R., Ricupero, N., Bucolo, C., Maugeri, F., Maltese, A., Puglisi, G. AAPS. PharmSciTech (2006)
- Enhancement of availability of cloricromene at brain level by a lipophilic prodrug. Pignatello, R., Maltese, A., Maugeri, F., Bucolo, C. J. Pharm. Pharmacol. (2006)
- Enhancement of drug affinity for cell membranes by conjugation with lipoamino acids. I. Synthesis and biological evaluation of lipophilic conjugates of tranylcypromine. Pignatello, R., Puleo, A., Guccione, S., Raciti, G., Acquaviva, R., Campisi, A., Ventura, C.A., Puglisi, G. Eur. J. Med. Chem (2005)
- Synthesis and in vitro skin permeation of naproxen conjugates with alpha-alkylamino acids. Pignatello, R., Montenegro, L., Stancampiano, A.H., Puleo, A., Puglisi, G. Current. Drug. Delivery (2005)
- Characterization of the mechanism of interaction in ibuprofen-Eudragit RL100 coevaporates. Pignatello, R., Spadaro, D., Vandelli, M.A., Forni, F., Puglisi, G. Drug. Dev. Ind. Pharm (2004)
- Lipophilic conjugates of methotrexate with short-chain alkylamino acids as DHFR inhibitors. Synthesis, biological evaluation, and molecular modeling. Pignatello, R., Guccione, S., Forte, S., Di Giacomo, C., Sorrenti, V., Vicari, L., Uccello Barretta, G., Balzano, F., Puglisi, G. Bioorg. Med. Chem. (2004)