Chemical Compound Review:
Acth (6-9) (2S)-2-[[(2S)-2-[[(2S)-2- amino-3-[4-[(2S)...
Synonyms:
AC1Q5DWV, AR-1F9084, AR-1F9085, AC1L4O63, 4289-02-5, ...
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- Structure-activity relationships of the melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH2 at the mouse melanocortin receptors. Part 3: modifications at the Arg position. Holder, J.R., Xiang, Z., Bauzo, R.M., Haskell-Luevano, C. Peptides (2003)
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- Activity and conformation of a cyclic heptapeptide possessing the message sequence His-Phe-Arg-Trp of alpha-melanotropin. Desai, P., Prachand, M., Coutinho, E., Saran, A., Bodi, J., Süli-Vargha, H. Int. J. Biol. Macromol. (2002)
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- Discovery of prototype peptidomimetic agonists at the human melanocortin receptors MC1R and MC4R. Haskell-Luevano, C., Hendrata, S., North, C., Sawyer, T.K., Hadley, M.E., Hruby, V.J., Dickinson, C., Gantz, I. J. Med. Chem. (1997)
- Synthesis and biological evaluation on hMC3, hMC4 and hMC5 receptors of gamma-MSH analogs substituted with L-alanine. Grieco, P., Balse-Srinivasan, P., Han, G., Weinberg, D., MacNeil, T., Van der Ploeg, L.H., Hruby, V.J. J. Pept. Res. (2002)
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