Chemical Compound Review:
Capromorelin 2-amino-N-[(2R)-1-[(1R)-1- benzyl-8-methyl...
Synonyms:
CHEMBL113313, SureCN1147592, CHEBI:282843, KST-1A2791, AC1Q5JMA, ...
Pan,
Carpino,
Lefker,
Ragan,
Toler,
Pettersen,
Nettleton,
Ng,
Pirie,
Chidsey-Frink,
Lu,
Nickerson,
Tess,
Mullins,
MacLean,
DaSilva-Jardine,
Thompson,
Carpino,
Lefker,
Toler,
Pan,
Hadcock,
Murray,
Cook,
DiBrino,
DeNinno,
Chidsey-Frink,
Hada,
Inthavongsay,
Lewis,
Mangano,
Mullins,
Nickerson,
Ng,
Pirie,
Ragan,
Rose,
Tess,
Wright,
Yu,
Zawistoski,
Pettersen,
DaSilva-Jardine,
Wilson,
Thompson,
Carpino,
Lefker,
Toler,
Pan,
Hadcock,
Cook,
DiBrino,
Campeta,
DeNinno,
Chidsey-Frink,
Hada,
Inthavongsay,
Mangano,
Mullins,
Nickerson,
Ng,
Pirie,
Ragan,
Rose,
Tess,
Wright,
Yu,
Zawistoski,
DaSilva-Jardine,
Wilson,
Thompson,
- Efficacy of a growth hormone-releasing peptide mimetic in cardiac ischemia/reperfusion injury. MacAndrew, J.T., Ellery, S.S., Parry, M.A., Pan, L.C., Black, S.C. Eur. J. Pharmacol. (2001)
- Gastric motor effects of peptide and non-peptide ghrelin agonists in mice in vivo and in vitro. Kitazawa, T., De Smet, B., Verbeke, K., Depoortere, I., Peeters, T.L. Gut (2005)
- Pyrazolinone-piperidine dipeptide growth hormone secretagogues (GHSs). Discovery of capromorelin. Carpino, P.A., Lefker, B.A., Toler, S.M., Pan, L.C., Hadcock, J.R., Cook, E.R., DiBrino, J.N., Campeta, A.M., DeNinno, S.L., Chidsey-Frink, K.L., Hada, W.A., Inthavongsay, J., Mangano, F.M., Mullins, M.A., Nickerson, D.F., Ng, O., Pirie, C.M., Ragan, J.A., Rose, C.R., Tess, D.A., Wright, A.S., Yu, L., Zawistoski, M.P., DaSilva-Jardine, P.A., Wilson, T.C., Thompson, D.D. Bioorg. Med. Chem. (2003)
- Discovery and biological characterization of capromorelin analogues with extended half-lives. Carpino, P.A., Lefker, B.A., Toler, S.M., Pan, L.C., Hadcock, J.R., Murray, M.C., Cook, E.R., DiBrino, J.N., DeNinno, S.L., Chidsey-Frink, K.L., Hada, W.A., Inthavongsay, J., Lewis, S.K., Mangano, F.M., Mullins, M.A., Nickerson, D.F., Ng, O., Pirie, C.M., Ragan, J.A., Rose, C.R., Tess, D.A., Wright, A.S., Yu, L., Zawistoski, M.P., Pettersen, J.C., DaSilva-Jardine, P.A., Wilson, T.C., Thompson, D.D. Bioorg. Med. Chem. Lett. (2002)
- Preclinical pharmacology of CP-424,391, an orally active pyrazolinone-piperidine [correction of pyrazolidinone-piperidine] growth hormone secretagogue. Pan, L.C., Carpino, P.A., Lefker, B.A., Ragan, J.A., Toler, S.M., Pettersen, J.C., Nettleton, D.O., Ng, O., Pirie, C.M., Chidsey-Frink, K., Lu, B., Nickerson, D.F., Tess, D.A., Mullins, M.A., MacLean, D.B., DaSilva-Jardine, P.A., Thompson, D.D. Endocrine (2001)