Chemical Compound Review:
CHEMBL327127 8-(2,6-dichlorophenyl)-3- [[3...
Synonyms:
SureCN256710, NSC-735424, DNC009907, NSC735424, PD-166326, ...
- PD166326, a novel tyrosine kinase inhibitor, has greater antileukemic activity than imatinib mesylate in a murine model of chronic myeloid leukemia. Wolff, N.C., Veach, D.R., Tong, W.P., Bornmann, W.G., Clarkson, B., Ilaria, R.L. Blood (2005)
- Caenorhabditis elegans ABL-1 antagonizes p53-mediated germline apoptosis after ionizing irradiation. Deng, X., Hofmann, E.R., Villanueva, A., Hobert, O., Capodieci, P., Veach, D.R., Yin, X., Campodonico, L., Glekas, A., Cordon-Cardo, C., Clarkson, B., Bornmann, W.G., Fuks, Z., Hengartner, M.O., Kolesnick, R. Nat. Genet. (2004)
- Activity of dual SRC-ABL inhibitors highlights the role of BCR/ABL kinase dynamics in drug resistance. Azam, M., Nardi, V., Shakespeare, W.C., Metcalf, C.A., Bohacek, R.S., Wang, Y., Sundaramoorthi, R., Sliz, P., Veach, D.R., Bornmann, W.G., Clarkson, B., Dalgarno, D.C., Sawyer, T.K., Daley, G.Q. Proc. Natl. Acad. Sci. U.S.A. (2006)
- A novel pyridopyrimidine inhibitor of abl kinase is a picomolar inhibitor of Bcr-abl-driven K562 cells and is effective against STI571-resistant Bcr-abl mutants. Huron, D.R., Gorre, M.E., Kraker, A.J., Sawyers, C.L., Rosen, N., Moasser, M.M. Clin. Cancer Res. (2003)