Chemical Compound Review:
Inogatran 2-[[(2R)-3-cyclohexyl-1- [(2S)-2-[3...
Synonyms:
SureCN22745, CHEMBL114715, SureCN871973, CHEBI:43313, CHEBI:288902, ...
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- Different mechanisms contribute to the biphasic pattern of carboxypeptidase U (TAFIa) generation during in vitro clot lysis in human plasma. Leurs, J., Wissing, B.M., Nerme, V., Schatteman, K., Björquist, P., Hendriks, D. Thromb. Haemost. (2003)
- BCH-2763, a novel potent parenteral thrombin inhibitor, is an effective antithrombotic agent in rodent models of arterial and venous thrombosis--comparisons with heparin, r-hirudin, hirulog, inogatran and argatroban. Finkle, C.D., St Pierre, A., Leblond, L., Deschenes, I., DiMaio, J., Winocour, P.D. Thromb. Haemost. (1998)
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- The effects of oral and intravenous direct thrombin inhibitors on the size of photochemically induced cortical infarction in rats. Mikulski, A., Elg, M., Gustafsson, D. Thromb. Res. (2001)
- Effects of inogatran, a new low-molecular-weight thrombin inhibitor, in rat models of venous and arterial thrombosis, thrombolysis and bleeding time. Gustafsson, D., Elg, M., Lenfors, S., Börjesson, I., Teger-Nilsson, A.C. Blood Coagul. Fibrinolysis (1996)
- Antithrombotic effect of LB-30057 (CI-1028), a new synthetic thrombin inhibitor, in a rabbit model of thrombosis: comparison with inogatran. Chi, L., Mertz, T.E., Rogers, K.L., Janiczek, N., Peng, Y.W., Saganek, L., Bousley, R.F., Juneau, P.L., Uprichard, A.C., Gallagher, K.P. J. Thromb. Thrombolysis (2001)
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- Population modelling of the effect of inogatran, at thrombin inhibitor, on ex vivo coagulation time (APTT) in healthy subjects and patients with coronary artery disease. Cullberg, M., Eriksson, U.G., Larsson, M., Karlsson, M.O. British journal of clinical pharmacology. (2001)
- Thrombin inhibition with inogatran for unstable angina pectoris: evidence for reactivated ischaemia after cessation of short-term treatment. Andersen, K., Dellborg, M., Emanuelsson, H., Grip, L., Swedberg, K. Coron. Artery Dis. (1996)
- Inhibition of endothelial cell-mediated generation of activated protein C by direct and antithrombin-dependent thrombin inhibitors. Linder, R., Frebelius, S., Jansson, K., Swedenborg, J. Blood Coagul. Fibrinolysis (2003)