Chemical Compound Review:
Delt-I (3S)-3-[[1-[[(1S)-1- (aminocarbonylmethylca...
Synonyms:
Deltorphin I, AC1L3XGS, LS-172539, C37H52N8O10, (D-Ala2)Deltorphin I, ...
- Differential sorting of human delta-opioid receptors after internalization by peptide and alkaloid agonists. Marie, N., Lecoq, I., Jauzac, P., Allouche, S. J. Biol. Chem. (2003)
- Met-enkephalin-containing peptides encoded by proenkephalin A mRNA expressed in activated murine thymocytes inhibit thymocyte proliferation. Linner, K.M., Quist, H.E., Sharp, B.M. J. Immunol. (1995)
- Neuropeptide FF (NPFF) analogs functionally antagonize opioid activities in NPFF2 receptor-transfected SH-SY5Y neuroblastoma cells. Mollereau, C., Mazarguil, H., Zajac, J.M., Roumy, M. Mol. Pharmacol. (2005)
- Helix-inducing alpha-aminoisobutyric acid in opioid mimetic deltorphin C analogues. Bryant, S.D., Guerrini, R., Salvadori, S., Bianchi, C., Tomatis, R., Attila, M., Lazarus, L.H. J. Med. Chem. (1997)
- Preparation and binding properties of radioiodinated analogues of dermorphin and deltorphin with high specificity for the mu- and delta-opioid receptors. Gaudriault, G., Zsürger, N., Vincent, J.P. J. Neurochem. (1997)
- Binding in vivo of selective mu and delta opioid agonists: localization by autoradiography. Mokhtari, M., Tafani, J.A., Zajac, J.M. Neuropeptides (1993)
- Binding to delta and mu opioid receptors by deltorphin I/II analogues modified at the Phe3 and Asp4/Glu4 side chains: a report of 32 new analogues and a QSAR study. Schullery, S.E., Mohammedshah, T., Makhlouf, H., Marks, E.L., Wilenkin, B.S., Escobar, S., Mousigian, C., Heyl, D.L. Bioorg. Med. Chem. (1997)
- Substitution of aromatic and nonaromatic amino acids for the Phe3 residue in the delta-selective opioid peptide deltorphin I: effects on binding affinity and selectivity. Heyl, D.L., Schmitter, S.J., Bouzit, H., Johnson, T.W., Hepp, A.M., Kurtz, K.R., Mousigian, C. Int. J. Pept. Protein Res. (1994)
- Activity of mu- and delta-opioid agonists in vas deferens from mice deficient in MOR gene. Maldonado, R., Severini, C., Matthes, H.W., Kieffer, B.L., Melchiorri, P., Negri, L. Br. J. Pharmacol. (2001)
- Transient expression of [D-Ala2] deltorphin I-like immunoreactivity in prenatal rat small intestine. Matsui, J., Fujimiya, M., Matsui, S., Amakata, Y., Renda, T., Kimura, H., Maeda, T. J. Histochem. Cytochem. (1994)
- Post-translational amino acid racemization in the frog skin peptide deltorphin I in the secretion granules of cutaneous serous glands. Auvynet, C., Seddiki, N., Dunia, I., Nicolas, P., Amiche, M., Lacombe, C. Eur. J. Cell Biol. (2006)
- Antinociceptive effects of isoleucine derivatives of deltorphin I and deltorphin II in rat spinal cord: a search for selectivity of delta receptor subtypes. Labuz, D., Toth, G., Machelska, H., Przewlocka, B., Borsodi, A., Przewłocki, R. Neuropeptides (1998)
- Fate of (D-Ala2)-deltorphin-I-like immunoreactive neurons in 6-hydroxydopamine lesioned rat brain. Casini, A., Pinna, A., Tooyama, I., Kimura, H., Di Chiara, G., Renda, T.G. European journal of histochemistry : EJH. (2004)
- Synthesis and biological properties of beta-MePhe3 analogues of deltorphin I and dermenkephalin: influence of biased chi 1 Phe3 residues on peptide recognition for delta-opioid receptors. Misicka, A., Cavagnero, S., Horvath, R., Davis, P., Porreca, F., Yamamura, H.I., Hruby, V.J. J. Pept. Res. (1997)
- Structure-activity relationships of dermorphin analogues containing N-substituted amino acids in the 2-position of the peptide sequence. Schmidt, R., Kálmán, A., Chung, N.N., Lemieux, C., Horváth, C., Schiller, P.W. Int. J. Pept. Protein Res. (1995)
- Phe3-substituted analogues of deltorphin C. Spatial conformation and topography of the aromatic ring in peptide recognition by delta opioid receptors. Salvadori, S., Bryant, S.D., Bianchi, C., Balboni, G., Scaranari, V., Attila, M., Lazarus, L.H. J. Med. Chem. (1993)
- A new selective antagonist of the nociceptin receptor. Guerrini, R., Calo, G., Rizzi, A., Bigoni, R., Bianchi, C., Salvadori, S., Regoli, D. Br. J. Pharmacol. (1998)
- Synthesis, conformation and biological activity of dermorphin and deltorphin I analogues containing N-alkylglycine in place of residues in position 1, 3, 5 and 6. Biondi, L., Giannini, E., Filira, F., Gobbo, M., Marastoni, M., Negri, L., Scolaro, B., Tomatisc, R., Rocchi, R. J. Pept. Sci. (2003)
- Dopamine depletion augments endogenous opioid-induced locomotion in the nucleus accumbens using both mu 1 and delta opioid receptors. Churchill, L., Roques, B.P., Kalivas, P.W. Psychopharmacology (Berl.) (1995)