Gene Review:
OPRM1 - opioid receptor, mu 1
Sus scrofa
- Dermorphin-related peptides from the skin of Phyllomedusa bicolor and their amidated analogs activate two mu opioid receptor subtypes that modulate antinociception and catalepsy in the rat. Negri, L., Erspamer, G.F., Severini, C., Potenza, R.L., Melchiorri, P., Erspamer, V. Proc. Natl. Acad. Sci. U.S.A. (1992)
- Comparison of mu opioid receptor binding on intact neuroblastoma cells with guinea pig brain and neuroblastoma cell membranes. Toll, L. J. Pharmacol. Exp. Ther. (1992)
- Chronic in utero morphine exposure alters mu-agonist-stimulated [35S]-GTPgammaS binding in neonatal and juvenile guinea pig brainstem regions associated with breathing control. Matsuda, A.Y., Olsen, G.D. Neurotoxicology and teratology. (2001)
- The molecular basis of opioid receptor function. Simonds, W.F. Endocr. Rev. (1988)
- Dual effect of trimebutine on contractility of the guinea pig ileum via the opioid receptors. Taniyama, K., Sano, I., Nakayama, S., Matsuyama, S., Takeda, K., Yoshihara, C., Tanaka, C. Gastroenterology (1991)
- Changes in opioid receptor selectivity following processing of peptide E: effect on gut motility. Davis, T.P., Gillespie, T.J., Shook, J., Kramer, T.H., Hoyer, G., Hawkins, K., Davis, P., Yamamura, H.I., Burks, T.F. Gastroenterology (1991)
- Agonist-selective endocytosis of mu opioid receptor by neurons in vivo. Sternini, C., Spann, M., Anton, B., Keith, D.E., Bunnett, N.W., von Zastrow, M., Evans, C., Brecha, N.C. Proc. Natl. Acad. Sci. U.S.A. (1996)
- The porcine mu opioid receptor: molecular cloning and mRNA distribution in lymphoid tissues. Pampusch, M.S., Osinski, M.A., Brown, D.R., Murtaugh, M.P. J. Neuroimmunol. (1998)
- Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Dooley, C.T., Chung, N.N., Schiller, P.W., Houghten, R.A. Proc. Natl. Acad. Sci. U.S.A. (1993)
- Design, synthesis, and biological activities of cyclic lactam peptide analogues of dynorphine A(1-11)-NH2. Lung, F.D., Collins, N., Stropova, D., Davis, P., Yamamura, H.I., Porreca, F., Hruby, V.J. J. Med. Chem. (1996)
- Synthesis and biological evaluation of 14-alkoxymorphinans. 2. (-)-N-(cyclopropylmethyl)-4,14-dimethoxymorphinan-6-one, a selective mu opioid receptor antagonist. Schmidhammer, H., Burkard, W.P., Eggstein-Aeppli, L., Smith, C.F. J. Med. Chem. (1989)
- Protein kinase A maintains cellular tolerance to mu opioid receptor agonists in hypothalamic neurosecretory cells with chronic morphine treatment: convergence on a common pathway with estrogen in modulating mu opioid receptor/effector coupling. Wagner, E.J., Rønnekleiv, O.K., Kelly, M.J. J. Pharmacol. Exp. Ther. (1998)
- Mu opioid receptor activation reduces inhibitory postsynaptic potentials in hippocampal CA3 pyramidal cells of rat and guinea pig. Caudle, R.M., Chavkin, C. J. Pharmacol. Exp. Ther. (1990)
- A comparison of the role of dynorphin in the hippocampal mossy fiber pathway in guinea pig and rat. Salin, P.A., Weisskopf, M.G., Nicoll, R.A. J. Neurosci. (1995)
- Modulation of G protein-coupled receptors by an estrogen receptor that activates protein kinase A. Lagrange, A.H., Ronnekleiv, O.K., Kelly, M.J. Mol. Pharmacol. (1997)
- Topographically designed analogues of [D-Pen,D-Pen5]enkephalin. Hruby, V.J., Toth, G., Gehrig, C.A., Kao, L.F., Knapp, R., Lui, G.K., Yamamura, H.I., Kramer, T.H., Davis, P., Burks, T.F. J. Med. Chem. (1991)
- Cyclic beta-casomorphin analogues with mixed mu agonist/delta antagonist properties: synthesis, pharmacological characterization, and conformational aspects. Schmidt, R., Vogel, D., Mrestani-Klaus, C., Brandt, W., Neubert, K., Chung, N.N., Lemieux, C., Schiller, P.W. J. Med. Chem. (1994)
- Subsensitivity to opioids is receptor-specific in isolated guinea pig ileum and mouse vas deferens after obstructive cholestasis. Dehpour, A.R., Rastegar, H., Jorjani, M., Roushanzamir, F., Joharchi, K., Ahmadiani, A. J. Pharmacol. Exp. Ther. (2000)
- Kappa opioid receptor tolerance in the guinea pig hippocampus. Jin, W., Terman, G.W., Chavkin, C. J. Pharmacol. Exp. Ther. (1997)
- N-methyl-D-aspartate receptors mediate endogenous opioid release in enteric neurons after abdominal surgery. Patierno, S., Zellalem, W., Ho, A., Parsons, C.G., Lloyd, K.C., Tonini, M., Sternini, C. Gastroenterology (2005)
- Sympathetic denervation-induced changes in G protein expression in enteric neurons of the guinea pig colon. Giaroni, C., Zanetti, E., Vanti, A., Canciani, L., Lecchini, S., Frigo, G. Life Sci. (2002)