Chemical Compound Review:
SureCN2141823 (2S)-N-[(1S)-1-[[(1S)-1- aminocarbonyl-3...
Synonyms:
GR-73632, LS-91361, AC1L3P3N, GR 73632, 133156-06-6
- What are the roles of substance P and neurokinin-1 receptors in the control of negative chronotropic or negative dromotropic vagal motoneurons? A physiological and ultrastructural analysis. Massari, V.J., Johnson, T.A., Gillis, R.A., Gatti, P.J. Brain Res. (1996)
- Ava[L-Pro9,N-MeLeu10] substance P(7-11) (GR 73632) and Sar9, Met(O2)11 increase distention-induced peristalsis through activation of neurokinin-1 receptors on smooth muscle and interstitial cells of cajal. Nieuwmeyer, F., Ye, J., Huizinga, J.D. J. Pharmacol. Exp. Ther. (2006)
- Centrally administered hemokinin-1 (HK-1), a neurokinin NK1 receptor agonist, produces substance P-like behavioral effects in mice and gerbils. Duffy, R.A., Hedrick, J.A., Randolph, G., Morgan, C.A., Cohen-Williams, M.E., Vassileva, G., Lachowicz, J.E., Laverty, M., Maguire, M., Shan, L.S., Gustafson, E., Varty, G.B. Neuropharmacology (2003)
- Pharmacological characterization of tachykinin NK2 receptors on isolated human urinary bladder, prostatic urethra and prostate. Palea, S., Corsi, M., Artibani, W., Ostardo, E., Pietra, C. J. Pharmacol. Exp. Ther. (1996)
- Effects of substance P on medial vestibular nucleus neurons in guinea-pig brainstem slices. Vibert, N., Serafin, M., Vidal, P.P., Muhlethaler, M. Eur. J. Neurosci. (1996)
- Increased ganglionic responses to substance P in hypertensive rats due to upregulation of NK(1) receptors. Schoborg, R.V., Hoover, D.B., Tompkins, J.D., Hancock, J.C. Am. J. Physiol. Regul. Integr. Comp. Physiol. (2000)
- Effects of TAK-637 on NK(1) receptor-mediated mechanisms regulating colonic secretion. Venkova, K., Greenwood-Van Meerveld, B. Toxicol. Appl. Pharmacol. (2004)
- Functional magnetic resonance mapping of intracerebroventricular infusion of a neuroactive peptide in the anaesthetised rat. Gozzi, A., Schwarz, A.J., Reese, T., Crestan, V., Bertani, S., Turrini, G., Corsi, M., Bifone, A. J. Neurosci. Methods (2005)
- Effect of the tachykinin NK1 receptor antagonists, RP 67580 and SR 140333, on electrically-evoked substance P release from rat spinal cord. Malcangio, M., Bowery, N.G. Br. J. Pharmacol. (1994)
- Chromodacryorrhea and repetitive hind paw tapping: models of peripheral and central tachykinin NK1 receptor activation in gerbils. Bristow, L.J., Young, L. Eur. J. Pharmacol. (1994)
- Characterization of substance P release from the intermediate area of rat thoracic spinal cord. Yang, L., Thomas, N.D., Helke, C.J. Synapse (1996)
- NK1 receptors in the medial hypothalamus potentiate defensive rage behavior elicited from the midbrain periaqueductal gray of the cat. Bhatt, S., Gregg, T.R., Siegel, A. Brain Res. (2003)