Chemical Compound Review:
Furamidine 4-[5-(4-carbamimidoylphenyl)- 2...
Synonyms:
Furandiamidine, CHEMBL24057, DB75, SureCN549198, AG-F-93517, ...
- Characterization of a novel DNA minor-groove complex. Nguyen, B., Hamelberg, D., Bailly, C., Colson, P., Stanek, J., Brun, R., Neidle, S., Wilson, W.D. Biophys. J. (2004)
- 3D QSAR on a library of heterocyclic diamidine derivatives with antiparasitic activity. Athri, P., Wenzler, T., Ruiz, P., Brun, R., Boykin, D.W., Tidwell, R., Wilson, W.D. Bioorg. Med. Chem. (2006)
- Distribution of furamidine analogues in tumor cells: targeting of the nucleus or mitochondria depending on the amidine substitution. Lansiaux, A., Tanious, F., Mishal, Z., Dassonneville, L., Kumar, A., Stephens, C.E., Hu, Q., Wilson, W.D., Boykin, D.W., Bailly, C. Cancer Res. (2002)
- Synthesis, DNA affinity, and antiprotozoal activity of linear dications: Terphenyl diamidines and analogues. Ismail, M.A., Arafa, R.K., Brun, R., Wenzler, T., Miao, Y., Wilson, W.D., Generaux, C., Bridges, A., Hall, J.E., Boykin, D.W. J. Med. Chem. (2006)
- Molecular determinants for DNA minor groove recognition: design of a bis-guanidinium derivative of ethidium that is highly selective for AT-rich DNA sequences. Bailly, C., Arafa, R.K., Tanious, F.A., Laine, W., Tardy, C., Lansiaux, A., Colson, P., Boykin, D.W., Wilson, W.D. Biochemistry (2005)
- Distribution of furamidine analogues in tumor cells: influence of the number of positive charges. Lansiaux, A., Dassonneville, L., Facompré, M., Kumar, A., Stephens, C.E., Bajic, M., Tanious, F., Wilson, W.D., Boykin, D.W., Bailly, C. J. Med. Chem. (2002)
- A crystallographic and spectroscopic study of the complex between d(CGCGAATTCGCG)2 and 2,5-bis(4-guanylphenyl)furan, an analogue of berenil. Structural origins of enhanced DNA-binding affinity. Laughton, C.A., Tanious, F., Nunn, C.M., Boykin, D.W., Wilson, W.D., Neidle, S. Biochemistry (1996)
- Dicationic diarylfurans as anti-Pneumocystis carinii agents. Boykin, D.W., Kumar, A., Spychala, J., Zhou, M., Lombardy, R.J., Wilson, W.D., Dykstra, C.C., Jones, S.K., Hall, J.E., Tidwell, R.R. J. Med. Chem. (1995)
- Unusual dehydroxylation of antimicrobial amidoxime prodrugs by cytochrome b5 and NADH cytochrome b5 reductase. Saulter, J.Y., Kurian, J.R., Trepanier, L.A., Tidwell, R.R., Bridges, A.S., Boykin, D.W., Stephens, C.E., Anbazhagan, M., Hall, J.E. Drug Metab. Dispos. (2005)
- Trypanocidal activity of the phenyl-substituted analogue of furamidine DB569 against Trypanosoma cruzi infection in vivo. de Souza, E.M., Oliveira, G.M., Boykin, D.W., Kumar, A., Hu, Q., De Nazaré C Soeiro, M. J. Antimicrob. Chemother. (2006)
- Trypanosoma rhodesiense: evaluation of the antitrypanosomal action of 2,5-bis(4-guanylphenyl)furan dihydrochloride. Steck, E.A., Kinnamon, K.E., Davidson, D.E., Duxbury, R.E., Johnson, A.J., Masters, R.E. Exp. Parasitol. (1982)
- Inhibition of HIV-1 Tat-TAR interaction by diphenylfuran derivatives: effects of the terminal basic side chains. Gelus, N., Bailly, C., Hamy, F., Klimkait, T., Wilson, W.D., Boykin, D.W. Bioorg. Med. Chem. (1999)