Chemical Compound Review:
Tocris-1709 9-methyl-3-[3- (trifluoromethyl)phenyl]- 1,2...
Synonyms:
CHEMBL13662, AG-G-51114, SureCN1320758, CHEBI:113358, CTK2F3997, ...
- CL 218,872 a triazolopyridazine with a selective affinity for the benzodiazepine BZ1 receptor subtype, retards the development and expression of amygdaloid-kindled seizures: effects of flumazenil. McNamara, R.K., Corcoran, M.E. Epilepsy Res. (1993)
- The separation of 3H-benzodiazepine binding sites in brain and of benzodiazepine pharmacological properties. Dubnick, B., Lippa, A.S., Klepner, C.A., Coupet, J., Greenblatt, E.N., Beer, B. Pharmacol. Biochem. Behav. (1983)
- The sedative effects of CL 218,872, like those of chlordiazepoxide, are reversed by benzodiazepine antagonists. File, S.E., Pellow, S., Wilks, L. Psychopharmacology (Berl.) (1985)
- Like diazepam, CL 218,872, a selective ligand for the benzodiazepine omega 1 receptor subtype, impairs place learning in the Morris water maze. McNamara, R.K., Skelton, R.W. Psychopharmacology (Berl.) (1992)
- Localization of type I benzodiazepine receptors to postsynaptic densities in bovine brain. Trifiletti, R.R., Snyder, S.H. J. Neurosci. (1985)
- In vivo binding of beta-carbolines in mice: regional differences and correlation of occupancy to pharmacological effects. Potier, M.C., Prado de Carvalho, L., Dodd, R.H., Besselievre, R., Rossier, J. Mol. Pharmacol. (1988)
- Development of benzodiazepine and picrotoxin (t-butylbicyclophosphorothionate) binding sites in rat cerebellar granule cells in culture. Squires, R.F., Saederup, E., Damgaard, I., Schousboe, A. J. Neurochem. (1990)
- Type I and type II gamma-aminobutyric acid/benzodiazepine receptors: purification and analysis of novel receptor complex from neonatal cortex. Sato, T.N., Neale, J.H. J. Neurochem. (1989)
- n-[3H]butyl-beta-carboline-3-carboxylate, a putative endogenous ligand, binds preferentially to subtype 1 of central benzodiazepine receptors. Medina, J.H., de Stein, M.L., De Robertis, E. J. Neurochem. (1989)
- Benzodiazepine-induced hyperphagia in the nondeprived rat: comparisons with CL 218,872, zopiclone, tracazolate and phenobarbital. Cooper, S.J., Moores, W.R. Pharmacol. Biochem. Behav. (1985)
- CL 218,872 binding to benzodiazepine receptors in rat spinal cord: modulation by gamma-aminobutyric acid and evidence for receptor heterogeneity. Villiger, J.W. J. Neurochem. (1984)
- Evidence for the presence of benzodiazepine receptor subclasses in different areas of the human brain. Montaldo, S., Serra, M., Concas, A., Corda, M.G., Mele, S., Biggio, G. Neurosci. Lett. (1984)
- Neurotransmitter receptors in the avian brain. III. GABA-benzodiazepine receptors. Dietl, M.M., Cortés, R., Palacios, J.M. Brain Res. (1988)
- The relationship of benzodiazepine binding sites to the norepinephrine projection in the hypothalamus of the adult rat. Harary, N., Kellogg, C. Brain Res. (1989)
- Effects of benzodiazepine receptor ligands on isolated rat superior cervical ganglia neurons. Aguayo, L.G., Cisternas, C., Tapia, J.C., Pancetti, F.C. Pharmacology (1996)
- Benzodiazepine receptor binding in young, mature and senescent rat brain and kidney. Pedigo, N.W., Schoemaker, H., Morelli, M., McDougal, J.N., Malick, J.B., Burks, T.F., Yamamura, H.I. Neurobiol. Aging (1981)
- Benzodiazepine receptor ligand actions on GABA responses. Benzodiazepines, CL 218872, zopiclone. Skerritt, J.H., Macdonald, R.L. Eur. J. Pharmacol. (1984)
- Modulation of [35S]TBPS binding by ligands with preferential affinity for benzodiazepine BZ1 sites in the cerebral cortex of newborn and adult rats. Giorgi, O., Lecca, D., Cancedda, E., Serra, G.P., Corda, M.G. Eur. J. Pharmacol. (1995)
- In vivo benzodiazepine receptor occupancy by CL 218,872 visualized by positron emission tomography in the brain of the living baboon: modulation by GABAergic transmission and relation with anticonvulsant activity. de la Sayette, V., Chavoix, C., Brouillet, E., Hantraye, P., Kunimoto, M., Khalili-Varasteh, M., Guibert, B., Prenant, C., Mazière, M. Experimental brain research. Experimentelle Hirnforschung. Expérimentation cérébrale. (1991)
- Benzodiazepine receptors increase in post-mortem brain of chronic schizophrenics. Kiuchi, Y., Kobayashi, T., Takeuchi, J., Shimizu, H., Ogata, H., Toru, M. European archives of psychiatry and neurological sciences. (1989)