Chemical Compound Review:
Tocris-1145 (2R,3S)-3-[[3,5- bis(trifluoromethyl)phenyl...
Synonyms:
CHEMBL27006, CHEBI:137245, CCG-204837, Lopac0_000752, DNC004178, ...
Muñoz,
Rosso,
Pérez,
Coveñas,
Rosso,
Zamarriego,
Piruat,
Muñoz,
Rosso,
Pérez,
Coveñas,
Rosso,
Zamarriego,
Soult,
Montero,
Langosch,
Kupferschmid,
Heinen,
Walden,
Herpfer,
Fiebich,
Lieb,
Rupniak,
Carlson,
Harrison,
Oates,
Seward,
Owen,
de Felipe,
Hunt,
Wheeldon,
Muñoz,
Pérez,
Coveñas,
Rosso,
Castro,
Varty,
Cohen-Williams,
Hunter,
Lieb,
Fiebich,
Herpfer,
Mantovani,
Löffler,
Feuerstein,
- Antitumoral action of the neurokinin-1-receptor antagonist L-733,060 and mitogenic action of substance P on human retinoblastoma cell lines. Muñoz, M., Rosso, M., Pérez, A., Coveñas, R., Rosso, R., Zamarriego, C., Soult, J.A., Montero, I. Invest. Ophthalmol. Vis. Sci. (2005)
- Neurokinin-1 (NK-1) receptor antagonists abrogate methamphetamine-induced striatal dopaminergic neurotoxicity in the murine brain. Yu, J., Cadet, J.L., Angulo, J.A. J. Neurochem. (2002)
- A general approach to (5S,6R)-6-alkyl-5-benzyloxy-2-piperidinones: application to the asymmetric syntheses of neurokinin substance P receptor antagonist (-)-L-733,061 and (-)-deoxocassine. Liu, L.X., Ruan, Y.P., Guo, Z.Q., Huang, P.Q. J. Org. Chem. (2004)
- The NK1 receptor is involved in the antitumoural action of L-733,060 and in the mitogenic action of substance P on neuroblastoma and glioma cell lines. Muñoz, M., Rosso, M., Pérez, A., Coveñas, R., Rosso, R., Zamarriego, C., Piruat, J.I. Neuropeptides (2005)
- Antitumoural action of L-733,060 on neuroblastoma and glioma cell lines. Muñoz, M., Pérez, A., Coveñas, R., Rosso, M., Castro, E. Archives italiennes de biologie. (2004)
- Enantioselective inhibition of the formalin paw late phase by the NK1 receptor antagonist L-733,060 in gerbils. Rupniak, N.M., Carlson, E., Boyce, S., Webb, J.K., Hill, R.G. Pain (1996)
- Endocannabinoids induce ileitis in rats via the capsaicin receptor (VR1). McVey, D.C., Schmid, P.C., Schmid, H.H., Vigna, S.R. J. Pharmacol. Exp. Ther. (2003)
- Pharmacological blockade or genetic deletion of substance P (NK(1)) receptors attenuates neonatal vocalisation in guinea-pigs and mice. Rupniak, N.M., Carlson, E.C., Harrison, T., Oates, B., Seward, E., Owen, S., de Felipe, C., Hunt, S., Wheeldon, A. Neuropharmacology (2000)
- Effects of substance P and its antagonist L-733060 on long term potentiation in guinea pig hippocampal slices. Langosch, J.M., Kupferschmid, S., Heinen, M., Walden, J., Herpfer, I., Fiebich, B.L., Lieb, K. Prog. Neuropsychopharmacol. Biol. Psychiatry (2005)
- No modulatory effect of neurokinin-1 receptor antagonists on serotonin uptake in human and rat brain synaptosomes. Lieb, K., Fiebich, B.L., Herpfer, I., Mantovani, M., Löffler, M., Feuerstein, T.J. European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology. (2005)
- Neurokinin receptors modulate the neurochemical actions of cocaine. Noailles, P.A., Angulo, J.A. Ann. N. Y. Acad. Sci. (2002)
- Substance P modulates cocaine-evoked dopamine overflow in the striatum of the rat brain. Kraft, M., Noailles, P., Angulo, J.A. Ann. N. Y. Acad. Sci. (2001)
- Ontogeny of neurokinin-1 receptor mediation of methamphetamine neurotoxicity in the striatum of the mouse brain. Yu, J., Allison, S., Ibrahim, D., Cadet, J.L., Angulo, J.A. Ann. N. Y. Acad. Sci. (2002)
- The antidepressant-like effects of neurokinin NK1 receptor antagonists in a gerbil tail suspension test. Varty, G.B., Cohen-Williams, M.E., Hunter, J.C. Behavioural pharmacology. (2003)
- Substance P and cholecystokinin regulate neurochemical responses to cocaine and methamphetamine in the striatum. Loonam, T.M., Noailles, P.A., Yu, J., Zhu, J.P., Angulo, J.A. Life Sci. (2003)
- L-733,060, a novel tachykinin NK1 receptor antagonist; effects in [Ca2+]i mobilisation, cardiovascular and dural extravasation assays. Seabrook, G.R., Shepheard, S.L., Williamson, D.J., Tyrer, P., Rigby, M., Cascieri, M.A., Harrison, T., Hargreaves, R.J., Hill, R.G. Eur. J. Pharmacol. (1996)