Chemical Compound Review:
Tocris-1808 N-[4-[[1-[2-(6-methylpyridin- 2-yl)ethyl]-4...
Synonyms:
CHEMBL327980, SureCN2168557, BSPBio_001313, KBioGR_000033, KBioSS_000033, ...
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- Class III antiarrhythmic drugs block HERG, a human cardiac delayed rectifier K+ channel. Open-channel block by methanesulfonanilides. Spector, P.S., Curran, M.E., Keating, M.T., Sanguinetti, M.C. Circ. Res. (1996)
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- Functional up-regulation of HERG K+ channels in neoplastic hematopoietic cells. Smith, G.A., Tsui, H.W., Newell, E.W., Jiang, X., Zhu, X.P., Tsui, F.W., Schlichter, L.C. J. Biol. Chem. (2002)
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- Expression and function of KCNH2 (HERG) in the human jejunum. Farrelly, A.M., Ro, S., Callaghan, B.P., Khoyi, M.A., Fleming, N., Horowitz, B., Sanders, K.M., Keef, K.D. Am. J. Physiol. Gastrointest. Liver Physiol. (2003)
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- Circadian changes of ether-a-go-go-related-gene (Erg) potassium channel transcripts in the rat pancreas and beta-cell. Mühlbauer, E., Bazwinsky, I., Wolgast, S., Klemenz, A., Peschke, E. Cell. Mol. Life Sci. (2007)
- Molecular and functional characterization of ERG, KCNQ, and KCNE subtypes in rat stomach smooth muscle. Ohya, S., Asakura, K., Muraki, K., Watanabe, M., Imaizumi, Y. Am. J. Physiol. Gastrointest. Liver Physiol. (2002)
- Autoimmunity against the second extracellular loop of beta(1)-adrenergic receptors induces early afterdepolarization and decreases in K-channel density in rabbits. Fukuda, Y., Miyoshi, S., Tanimoto, K., Oota, K., Fujikura, K., Iwata, M., Baba, A., Hagiwara, Y., Yoshikawa, T., Mitamura, H., Ogawa, S. J. Am. Coll. Cardiol. (2004)
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