Chemical Compound Review:
DISOXARIL 5-[7-[4-(4,5-dihydro-1,3- oxazol-2...
Synonyms:
Disoxarilo, Disoxarilum, Compound IV, CHEMBL283639, SureCN147146, ...
- The site of attachment in human rhinovirus 14 for antiviral agents that inhibit uncoating. Smith, T.J., Kremer, M.J., Luo, M., Vriend, G., Arnold, E., Kamer, G., Rossmann, M.G., McKinlay, M.A., Diana, G.D., Otto, M.J. Science (1986)
- Distribution of drug resistance mutations in type 3 poliovirus identifies three regions involved in uncoating functions. Mosser, A.G., Sgro, J.Y., Rueckert, R.R. J. Virol. (1994)
- WIN 51711-dependent mutants of poliovirus type 3: evidence that virions decay after release from cells unless drug is present. Mosser, A.G., Rueckert, R.R. J. Virol. (1993)
- In vitro activity of WIN 51711, a new broad-spectrum antipicornavirus drug. Otto, M.J., Fox, M.P., Fancher, M.J., Kuhrt, M.F., Diana, G.D., McKinlay, M.A. Antimicrob. Agents Chemother. (1985)
- Use of WIN 51711 to prevent echovirus type 9-induced paralysis in suckling mice. McKinlay, M.A., Frank, J.A., Benziger, D.P., Steinberg, B.A. J. Infect. Dis. (1986)
- Anticonvulsant activities of 4-bromobenzaldehyde semicarbazone. Dimmock, J.R., Baker, G.B. Epilepsia (1994)
- Difluorothromboxane A2 and stereoisomers: stable derivatives of thromboxane A2 with differential effects on platelets and blood vessels. Morinelli, T.A., Okwu, A.K., Mais, D.E., Halushka, P.V., John, V., Chen, C.K., Fried, J. Proc. Natl. Acad. Sci. U.S.A. (1989)
- Structure determination of antiviral compound SCH 38057 complexed with human rhinovirus 14. Zhang, A., Nanni, R.G., Li, T., Arnold, G.F., Oren, D.A., Jacobo-Molina, A., Williams, R.L., Kamer, G., Rubenstein, D.A., Li, Y. J. Mol. Biol. (1993)
- Inhibitors of poliovirus uncoating efficiently block the early membrane permeabilization induced by virus particles. Almela, M.J., González, M.E., Carrasco, L. J. Virol. (1991)
- Two groups of rhinoviruses revealed by a panel of antiviral compounds present sequence divergence and differential pathogenicity. Andries, K., Dewindt, B., Snoeks, J., Wouters, L., Moereels, H., Lewi, P.J., Janssen, P.A. J. Virol. (1990)
- Prevention of rhinovirus and poliovirus uncoating by WIN 51711, a new antiviral drug. Fox, M.P., Otto, M.J., McKinlay, M.A. Antimicrob. Agents Chemother. (1986)
- A comparison of WIN 51711 and R 78206 as stabilizers of poliovirus virions and procapsids. Rombaut, B., Andries, K., Boeyé, A. J. Gen. Virol. (1991)
- Potent and selective inhibitors of leukotriene A4 hydrolase: effects on purified enzyme and human polymorphonuclear leukocytes. Wetterholm, A., Haeggström, J.Z., Samuelsson, B., Yuan, W., Munoz, B., Wong, C.H. J. Pharmacol. Exp. Ther. (1995)
- Anti-inflammatory effects and mechanisms of the ethanol extract of Evodia rutaecarpa and its bioactive components on neutrophils and microglial cells. Ko, H.C., Wang, Y.H., Liou, K.T., Chen, C.M., Chen, C.H., Wang, W.Y., Chang, S., Hou, Y.C., Chen, K.T., Chen, C.F., Shen, Y.C. Eur. J. Pharmacol. (2007)
- Effects of some pyrrolic and dihydropyrrolizine esters on mouse skin: a preliminary study. Mattocks, A.R., Cabral, J.R. Tumori. (1979)
- Rapid release of an alpha-adrenergic receptor ligand from photolabile analogues. Walker, J.W., Martin, H., Schmitt, F.R., Barsotti, R.J. Biochemistry (1993)
- 3-[4'-bromo-(1,1'-biphenyl)-4-yl]-N, N-dimethyl-3-(2-thienyl)-2-propen-1-amine: synthesis, cytotoxicity, and leishmanicidal, trypanocidal and antimycobacterial activities. de Souza, A.O., Hemerly, F.P., Busollo, A.C., Melo, P.S., Machado, G.M., Miranda, C.C., Santa-Rita, R.M., Haun, M., Leon, L.L., Sato, D.N., de Castro, S.L., Durán, N. J. Antimicrob. Chemother. (2002)
- Inhibition of poliovirus uncoating by disoxaril (WIN 51711). Zeichhardt, H., Otto, M.J., McKinlay, M.A., Willingmann, P., Habermehl, K.O. Virology (1987)
- Location of the sulphonylurea receptor at the cytoplasmic face of the beta-cell membrane. Schwanstecher, M., Schwanstecher, C., Dickel, C., Chudziak, F., Moshiri, A., Panten, U. Br. J. Pharmacol. (1994)
- Ionization characteristics of the Cys-25/His-159 interactive system and of the modulatory group of papain: resolution of ambiguity by electronic perturbation of the quasi-2-mercaptopyridine leaving group in a new pyrimidyl disulphide reactivity probe. Mellor, G.W., Thomas, E.W., Topham, C.M., Brocklehurst, K. Biochem. J. (1993)
- Analysis of the antagonistic actions of HOE 140 and other novel bradykinin analogues on the guinea-pig ileum. Griesbacher, T., Lembeck, F. Eur. J. Pharmacol. (1992)
- Preparation and characterization of S-[2-carboxy-1-(1H-imidazol-4-yl)ethyl]glutathione and its derivatives as proposed precursors of S-[2-carboxy-1-(1H-imidazol-4-yl)ethyl]cysteine, a compound found in human urine. Kinuta, M., Ubuka, T., Yao, K., Yamada, S., Yukihiro, K., Tomozawa, M. Biochim. Biophys. Acta (1993)
- Synthesis and cytotoxicity of platinum(II) complexes of 3-aminocyclopentanespiro-5-hydantoin and 3-aminocycloheptanespiro-5-hydantoin. Kushev, D., Naydenova, E., Popova, J., Maneva, L., Grancharov, K., Spassovska, N. Z. Naturforsch., C, J. Biosci. (2003)
- The renal action of spirorenone and other 6 beta,7 beta; 15 beta,16 beta-dimethylene-17-spirolactones, a new type of steroidal aldosterone antagonists. Casals-Stenzel, J., Buse, M., Wambach, G., Losert, W. Arzneimittel-Forschung. (1984)
- In vivo distribution studies of radioactively labelled platinum complexes; cis-dichlorodiammine platinum(II), cis-trans-dichlorodihydroxy-bis-(isopropylamine) platinum(IV), cis-dichloro-bis-cyclopropylamine platinum(II), and cis-diammine 1,1-cyclobutanedicarboxylate platinum(II) in patients with malignant disease, using a gamma camera. Owens, S.E., Thatcher, N., Sharma, H., Adam, N., Harrison, R., Smith, A., Zaki, A., Baer, J.C., McAuliffe, C.A., Crowther, D. Cancer Chemother. Pharmacol. (1985)
- Thermal degradation products formed from carotenoids during a heat-induced degradation process of paprika oleoresins (Capsicum annuum L.). Pérez-Gálvez, A., Rios, J.J., Mínguez-Mosquera, M.I. J. Agric. Food Chem. (2005)
- Non-benzodiazepine anxiolytics: potential activity of phenylpiperazines without 3H-diazepam displacing action. Lloyd, K.G., Depoortere, H., Scatton, B., Schoemaker, H., Zivkovic, B., Manoury, P., Langer, S.Z., Morselli, P.L., Bartholini, G. Pharmacol. Biochem. Behav. (1985)