Chemical Compound Review:
Redeptin 8-[4,4-bis(4- fluorophenyl)butyl]-1- phenyl...
Synonyms:
Fluspirilen, Fluspirilene, Fluspirileno, Imap, Fluspirilenum, ...
- A controlled clinical trial of fluspirilene, a long-acting injectable neuroleptic, in schizophrenic patients with acute exacerbation. Chouinard, G., Annable, L., Steinberg, S. Journal of clinical psychopharmacology. (1986)
- Safety of long-term neuroleptanxiolysis with fluspirilene 1.5 mg per week. Tegeler, J., Lehmann, E., Weiher, A., Heinrich, K. Pharmacopsychiatry (1990)
- Dystonic dysphagia associated with fluspirilene. Stones, M., Kennie, D.C., Fulton, J.D. BMJ (1990)
- Depot fluspirilene for schizophrenia. Abhijnhan, A., Adams, C., David, A., Ozbilen, M. Cochrane database of systematic reviews (Online) (2007)
- Test therapy in the treatment of generalized anxiety disorders with low dose fluspirilene. Wurthmann, C., Klieser, E., Lehmann, E., Pester, U. Prog. Neuropsychopharmacol. Biol. Psychiatry (1995)
- Antischizophrenic drugs of the diphenylbutylpiperidine type act as calcium channel antagonists. Gould, R.J., Murphy, K.M., Reynolds, I.J., Snyder, S.H. Proc. Natl. Acad. Sci. U.S.A. (1983)
- Blockade of low and high threshold Ca2+ channels by diphenylbutylpiperidine antipsychotics linked to inhibition of prolactin gene expression. Enyeart, J.J., Biagi, B.A., Day, R.N., Sheu, S.S., Maurer, R.A. J. Biol. Chem. (1990)
- Substituted diphenylbutylpiperidines bind to a unique high affinity site on the L-type calcium channel. Evidence for a fourth site in the cardiac calcium entry blocker receptor complex. King, V.F., Garcia, M.L., Shevell, J.L., Slaughter, R.S., Kaczorowski, G.J. J. Biol. Chem. (1989)
- Preferential block of T-type calcium channels by neuroleptics in neural crest-derived rat and human C cell lines. Enyeart, J.J., Biagi, B.A., Mlinar, B. Mol. Pharmacol. (1992)
- Inhibition of synaptic transmission and epileptiform activity in central neurones by fluspirilene. Wang, S.J., Lu, K.T., Gean, P.W. Br. J. Pharmacol. (1997)
- A six-month follow-up of refractory chronic psychotics treated with Haldol-AID. Wouters, J. Acta psychiatrica Belgica. (1978)
- Choline high-affinity uptake and metabolism and choline acetyltransferase activity in the striatum of rats chronically treated with neuroleptics. Pedata, F., Sorbi, S., Pepeu, G. J. Neurochem. (1980)
- Selective antagonism of calcium channel activators by fluspirilene. Kenny, B.A., Fraser, S., Kilpatrick, A.T., Spedding, M. Br. J. Pharmacol. (1990)
- Fluspirilene block of N-type calcium current in NGF-differentiated PC12 cells. Grantham, C.J., Main, M.J., Cannell, M.B. Br. J. Pharmacol. (1994)
- Risperidone compared with new and reference antipsychotic drugs: in vitro and in vivo receptor binding. Schotte, A., Janssen, P.F., Gommeren, W., Luyten, W.H., Van Gompel, P., Lesage, A.S., De Loore, K., Leysen, J.E. Psychopharmacology (Berl.) (1996)
- Abscisic acid plasmalemma perception triggers a calcium influx essential for RAB18 gene expression in Arabidopsis thaliana suspension cells. Ghelis, T., Dellis, O., Jeannette, E., Bardat, F., Miginiac, E., Sotta, B. FEBS Lett. (2000)
- Inhibition of glutamate release by fluspirilene in cerebrocortical nerve terminals (synaptosomes). Wang, S.J. Synapse (2002)
- The role of Ca2+ channels of the L-type in neurotransmitter plasticity of cultured sympathetic neurons. Vidal, S., Raynaud, B., Weber, M.J. Brain Res. Mol. Brain Res. (1989)
- Induction of the vesicular monoamine transporter by elevated potassium concentration in cultures of rat sympathetic neurons. Desnos, C., Raynaud, B., Vidal, S., Weber, M.J., Scherman, D. Brain Res. Dev. Brain Res. (1990)
- Fluspirilene (Imap) in the treatment of psychosomatic complaints in hypochondriacal patients. Kalis, D., Ten Oever, G.H., Erdmann, J.F. Acta psychiatrica Belgica. (1980)
- Unilateral deep brain stimulation of the internal globus pallidus alleviates tardive dyskinesia. Schrader, C., Peschel, T., Petermeyer, M., Dengler, R., Hellwig, D. Mov. Disord. (2004)
- A retrospective evaluation of long-term fluspirilene (IMAP) treatment. Tanghe, A. Acta psychiatrica Belgica. (1976)