Chemical Compound Review:
CHEMBL285755 7-(dipropylamino)-5,6,7,8...
Synonyms:
SureCN623950, AG-J-78903, DP-7-AT, CHEBI:152338, CCG-204705, ...
- S33084, a novel, potent, selective, and competitive antagonist at dopamine D(3)-receptors: II. Functional and behavioral profile compared with GR218,231 and L741,626. Millan, M.J., Dekeyne, A., Rivet, J.M., Dubuffet, T., Lavielle, G., Brocco, M. J. Pharmacol. Exp. Ther. (2000)
- Mechanisms and sites of ocular action of 7-hydroxy-2-dipropylaminotetralin: a dopamine(3) receptor agonist. Chu, E., Chu, T.C., Potter, D.E. J. Pharmacol. Exp. Ther. (2000)
- Involvement of dopamine D3 receptors in the area postrema in R(+)-7-OH-DPAT-induced emesis in the ferret. Yoshikawa, T., Yoshida, N., Hosoki, K. Eur. J. Pharmacol. (1996)
- Effects of putative dopamine D3 receptor agonists, 7-OH-DPAT, and quinpirole, on yawning, stereotypy, and body temperature in rats. Kurashima, M., Yamada, K., Nagashima, M., Shirakawa, K., Furukawa, T. Pharmacol. Biochem. Behav. (1995)
- Additive hypothermic effects of the 5-HT1A receptor agonist 8-OH-DPAT and the dopamine D2/3 receptor agonist 7-OH-DPAT in the rat. Eltayb, A., Lindblom, S., Oerther, S., Ahlenius, S. Acta Physiol. Scand. (2001)
- Differential effects of 7-OH-DPAT and apomorphine on hyperactivity induced by MK-801 (dizocilpine) in rats. Clements, R.L., Greenshaw, A.J. Neuropharmacology (2005)
- Local administration of dopaminergic drugs into the ventral tegmental area modulates cataplexy in the narcoleptic canine. Reid, M.S., Tafti, M., Nishino, S., Sampathkumaran, R., Siegel, J.M., Mignot, E. Brain Res. (1996)
- The dopamine receptor agonist 7-OH-DPAT modulates the acquisition and expression of morphine-induced place preference. Rodríguez De Fonseca, F., Rubio, P., Martín-Calderón, J.L., Caine, S.B., Koob, G.F., Navarro, M. Eur. J. Pharmacol. (1995)
- Investigations into the nature of a 7-OH-DPAT discriminative cue: comparison with D-amphetamine. Varty, G.B., Higgins, G.A. Eur. J. Pharmacol. (1997)
- The putative dopamine D3 agonist, 7-OH-DPAT, reduces dopamine release in the nucleus accumbens and electrical self-stimulation to the ventral tegmentum. Gilbert, D.B., Millar, J., Cooper, S.J. Brain Res. (1995)
- Modulation of cocaine self-administration in the rat through D-3 dopamine receptors. Caine, S.B., Koob, G.F. Science (1993)
- Psychostimulant-induced Fos protein expression in the thalamic paraventricular nucleus. Deutch, A.Y., Bubser, M., Young, C.D. J. Neurosci. (1998)
- Dopamine D(3) receptors and salt-dependent hypertension. Luippold, G., Zimmermann, C., Mai, M., Kloor, D., Starck, D., Gross, G., Mühlbauer, B. J. Am. Soc. Nephrol. (2001)
- Gialpha3 protein-coupled dopamine D3 receptor-mediated inhibition of renal NHE3 activity in SHR proximal tubular cells is a PLC-PKC-mediated event. Pedrosa, R., Gomes, P., Hopfer, U., Jose, P.A., Soares-da-Silva, P. Am. J. Physiol. Renal Physiol. (2004)
- 7-OH-DPAT and PD 128907 selectively activate the D3 dopamine receptor in a novel environment. Pritchard, L.M., Logue, A.D., Hayes, S., Welge, J.A., Xu, M., Zhang, J., Berger, S.P., Richtand, N.M. Neuropsychopharmacology (2003)
- Bromocriptine and quinpirole, but not 7-OH-DPAT or SKF 38393, potentiate the inhibitory effect of L-NAME on ethanol-induced locomotor activity in mice. Uzbay, I.T., Kayir, H. Naunyn Schmiedebergs Arch. Pharmacol. (2003)
- Independent roles of dopamine D1 and D2/3 receptors in rat thermoregulation. Salmi, P. Brain Res. (1998)
- Postglomerular vasoconstriction induced by dopamine D(3) receptor activation in anesthetized rats. Luippold, G., Schneider, S., Vallon, V., Osswald, H., Mühlbauer, B. Am. J. Physiol. Renal Physiol. (2000)
- Behavioral effects induced by the dopamine D3 agonist 7-OH-DPAT in sexually-active and -inactive male rats. Ferrari, F., Giuliani, D. Neuropharmacology (1996)
- The dopamine D3/2 agonist 7-OH-DPAT attenuates the development of morphine tolerance but not physical dependence in rats. Cook, C.D., Barrett, A.C., Syvanthong, C., Picker, M.J. Psychopharmacology (Berl.) (2000)
- Increased levels of proneurotensin/neuromedin N mRNA in rat striatum and nucleus accumbens induced by 7-OH-DPAT and nafadotride. Levant, B., Garimelli, B., Shafer, R.A., Merchant, K.M. Neuropsychopharmacology (1999)
- Differential regulation of dopamine D2 and D3 receptors by chronic drug treatments. Stanwood, G.D., Lucki, I., McGonigle, P. J. Pharmacol. Exp. Ther. (2000)
- D2 dopamine receptors and modulation of spontaneous acetylcholine (ACh) release from rat striatal synaptosomes. Clos, M.V., García-Sanz, A., Vivas, N.M., Badia, A. Br. J. Pharmacol. (1997)
- Presynaptic dopamine autoreceptors control tyrosine hydroxylase activation in depolarized striatal dopaminergic terminals. el Mestikawy, S., Glowinski, J., Hamon, M. J. Neurochem. (1986)
- C1- and C3-methyl-substituted derivatives of 7-hydroxy-2-(di-n-propylamino)tetralin: activities at central dopamine receptors. Johansson, A.M., Nilsson, J.L., Karlén, A., Hacksell, U., Sanchez, D., Svensson, K., Hjorth, S., Carlsson, A., Sundell, S., Kenne, L. J. Med. Chem. (1987)
- Discriminative stimulus properties of the dopamine D3 receptor agonists, PD128,907 and 7-OH-DPAT: a comparative characterization with novel ligands at D3 versus D2 receptors. Millan, M.J., Girardon, S., Monneyron, S., Dekeyne, A. Neuropharmacology (2000)
- Interactions of (+)- and (-)-8- and 7-hydroxy-2-(di-n-propylamino)tetralin at human (h)D3, hD2 and h serotonin1A receptors and their modulation of the activity of serotoninergic and dopaminergic neurones in rats. Lejeune, F., Newman-Tancredi, A., Audinot, V., Millan, M.J. J. Pharmacol. Exp. Ther. (1997)
- Characterization of the human dopamine D3 receptor expressed in transfected cell lines. MacKenzie, R.G., VanLeeuwen, D., Pugsley, T.A., Shih, Y.H., Demattos, S., Tang, L., Todd, R.D., O'Malley, K.L. Eur. J. Pharmacol. (1994)
- Effects of selective serotonin and dopamine agonists on plasma levels of glucose, insulin and glucagon in the rat. Uvnäs-Moberg, K., Ahlenius, S., Alster, P., Hillegaart, V. Neuroendocrinology (1996)
- Biphasic effects of D3-receptor agonists, 7-OH-DPAT and PD128907, on the D1-receptor agonist-induced hyperactivity in mice. Mori, T., Murase, K., Tanaka, J., Ichimaru, Y. Jpn. J. Pharmacol. (1997)
- Dopamine D2 receptor knock-out mice are insensitive to the hypolocomotor and hypothermic effects of dopamine D2/D3 receptor agonists. Boulay, D., Depoortere, R., Perrault, G., Borrelli, E., Sanger, D.J. Neuropharmacology (1999)
- Alterations in dopamine D3 receptors in the circling (ci3) rat mutant. Schirmer, M., Nobrega, J.N., Harrison, S.J., Löscher, W. Neuroscience (2007)
- Estimation of the interstitial free concentration of the putative dopamine D3 receptor selective agonist 7-OH-DPAT in the dorsal striatum of freely moving rats. Gainetdinov, R.R., Sotnikova, T.D., Grekhova, T.V., Rayevsky, K.S. Neurosci. Lett. (1995)
- Effects of (-)eticlopride and 7-OH-DPAT on the tail-suspension test in mice. Ferrari, F., Giuliani, D. J. Psychopharmacol. (Oxford) (1997)