Chemical Compound Review:
tiapride N-(2-diethylaminoethyl)-2- methoxy-5...
Synonyms:
Tiaprida, Thiapride, Tiapridal, Tiapridum, Lopac-T-0410, ...
Kotzailias,
Finsterer,
Aull,
Eichler,
Pratscher,
Jilma,
Lucht,
Kuehn,
Schroeder,
Armbruster,
Abraham,
Schattenberg,
Gaensicke,
Barnow,
Tretzel,
Herrmann,
Freyberger,
- Tiapride in Parkinson's disease. Price, P., Parkes, J.D., Marsden, C.D. Lancet (1978)
- Tiapride-induced torsade de pointes. Iglesias, E., Esteban, E., Zabala, S., Gascon, A. Am. J. Med. (2000)
- Tiapride in the treatment of tardive dyskinesia: a clinical and biochemical study. Perényi, A., Arató, M., Bagdy, G., Frecska, E., Szücs, R. The Journal of clinical psychiatry. (1985)
- Tiapride. A review of its pharmacology and therapeutic potential in the management of alcohol dependence syndrome. Peters, D.H., Faulds, D. Drugs (1994)
- Effects of tiapride in tardive dyskinesia. Pollak, P., Gaio, J.M., Hommel, M., Pellat, J., Perret, J. Psychopharmacology (Berl.) (1985)
- Cataplexy relieved by tiapride. Paulus, W., Hömberg, V., Noth, J. Arch. Neurol. (1983)
- Tiapride in the prevention of relapse in recently detoxified alcoholics. Shaw, G.K., Waller, S., Majumdar, S.K., Alberts, J.L., Latham, C.J., Dunn, G. The British journal of psychiatry : the journal of mental science. (1994)
- Tiapride in 12 Huntington's disease patients. Quinn, N., Marsden, C.D. J. Neurol. Neurosurg. Psychiatr. (1985)
- Involvement of dopaminergic neurotransmission in the control of goal-directed movements. Schmidt, W.J. Psychopharmacology (Berl.) (1983)
- Measuring the efficacy of psychopharmacological treatment of psychomotoric restlessness in dementia: clinical evaluation of tiapride. Gutzmann, H., Kühl, K.P., Kanowski, S., Khan-Boluki, J. Pharmacopsychiatry (1997)
- Influence of the dopamine D2 receptor (DRD2) exon 8 genotype on efficacy of tiapride and clinical outcome of alcohol withdrawal. Lucht, M.J., Kuehn, K.U., Schroeder, W., Armbruster, J., Abraham, G., Schattenberg, A., Gaensicke, M., Barnow, S., Tretzel, H., Herrmann, F.H., Freyberger, H.J. Pharmacogenetics (2001)
- Prediction of catalepsies induced by amiodarone, aprindine and procaine: similarity in conformation of diethylaminoethyl side chain. Matsui, A., Matsuo, H., Takanaga, H., Sasaki, S., Maeda, M., Sawada, Y. J. Pharmacol. Exp. Ther. (1998)
- Functional analysis of the D2L dopamine receptor expressed in a cAMP-responsive luciferase reporter cell line. George, S.E., Bungay, P.J., Naylor, L.H. Biochem. Pharmacol. (1998)
- Differential regulation of D2 and D4 dopamine receptor mRNAs in the primate cerebral cortex vs. neostriatum: effects of chronic treatment with typical and atypical antipsychotic drugs. Lidow, M.S., Goldman-Rakic, P.S. J. Pharmacol. Exp. Ther. (1997)
- Down-regulation of the D1 and D5 dopamine receptors in the primate prefrontal cortex by chronic treatment with antipsychotic drugs. Lidow, M.S., Elsworth, J.D., Goldman-Rakic, P.S. J. Pharmacol. Exp. Ther. (1997)
- L-dopa-induced respiratory disturbance in Parkinson's disease suppressed by tiapride. De Keyser, J., Vincken, W. Neurology (1985)
- The benzamide tiapride: treatment of extrapyramidal motor and other clinical syndromes. Dose, M., Lange, H.W. Pharmacopsychiatry (2000)
- Tourette syndrome: efficient treatment with ziprasidone and normalization of body weight in a patient with excessive weight gain under tiapride. Meisel, A., Winter, C., Zschenderlein, R., Arnold, G. Mov. Disord. (2004)
- Early administration of tiapride to young rats without long-lasting changes in the development of the dopaminergic system. Bock, N., Moll, G.H., Wicker, M., Pilz, J., Rüther, E., Banaschewski, T., Huether, G., Rothenberger, A. Pharmacopsychiatry (2004)
- Comparative study of tiapride and neuroleptics with anti-dopamine activity on convulsive seizure in mice. Satoh, H., Nakanishi, H., Shirakawa, K., Kohjimoto, Y., Kuwaki, T., Ono, T., Shibayama, F. Jpn. J. Pharmacol. (1987)
- Influence of tiapride on platelet counts in healthy volunteers and patients with movement disorders. Kotzailias, N., Finsterer, J., Aull, S., Eichler, H.G., Pratscher, B., Jilma, B. Prog. Neuropsychopharmacol. Biol. Psychiatry (2003)
- Single oral dose pharmacokinetics of tiapride in patients with Huntington's disease. Norman, T., Chiu, E., James, R.H., Gregory, M.S. Eur. J. Clin. Pharmacol. (1987)
- Tiapride. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in geriatric agitation. Steele, J.W., Faulds, D., Sorkin, E.M. Drugs & aging. (1993)
- Comparison of effects of tiapride and sulpiride on D-1, D-2, D-3 and D-4 subtypes of dopamine receptors in rat striatal and bovine caudate nucleus membranes. Arima, T., Samura, N., Nomura, Y., Segawa, T. Jpn. J. Pharmacol. (1986)
- Tiapride-induced chronic hyperprolactinaemia: interference with the human menstrual cycle. L'Hermite, M., Michaux-Duchêne, A., Robyn, C. Acta Endocrinol. (1979)
- Benzamide action at alpha 2-adrenoceptors modifies catecholamine-induced contraction and relaxation of circular smooth muscle from guinea-pig stomach. Sahyoun, H.A., Costall, B., Naylor, R.J. Naunyn Schmiedebergs Arch. Pharmacol. (1982)
- Effects of tiapride infusion on plasma levels of beta-endorphin, prolactin and dopamine in patients with pain from cancer. Gennari, C., Nami, R., Pizzuti, M., D'Ascenzo, G., Bianchini, C. Pathol. Biol. (1981)
- Effect of tiapride on electroacupuncture analgesia. Dai, J.L., Xu, S.F. Zhongguo yao li xue bao = Acta pharmacologica Sinica. (1991)
- Acute dyskinesias in monkeys elicited by halopemide, mezilamine and the "antidyskinetic" drugs, oxiperomide and tiapride. Neale, R., Fallon, S., Gerhardt, S., Liebman, J.M. Psychopharmacology (Berl.) (1981)
- Tiapride attenuates pain transmission through an indirect activation of central serotonergic mechanism. Takeshita, N., Ohkubo, Y., Yamaguchi, I. J. Pharmacol. Exp. Ther. (1995)
- Determination of sultopride and tiapride in serum by gas chromatography using a surface ionisation detector. Kamizono, A., Inotsume, N., Miyamoto, K., Ueda, K., Miyakawa, T., Arimoto, H., Nakano, M. J. Chromatogr. (1991)
- Treatment of alcohol withdrawal: tiapride and carbamazepine versus clomethiazole. A pilot study. Franz, M., Dlabal, H., Kunz, S., Ulferts, J., Gruppe, H., Gallhofer, B. European archives of psychiatry and clinical neuroscience. (2001)
- Effects of tiapride on homovanillic acid levels in human cerebrospinal fluid drawn at pneumoencephalography. Spissu, A., Congia, S., Piccardi, M.P., Fadda, F., Mangoni, A., Gessa, G.L. Psychopharmacology (Berl.) (1980)
- Tiapride: effects on tardive dyskinesia and on prolactin plasma concentrations. Greil, W., Auberger, S., Haag, H., Rüther, E. Neuropsychobiology (1985)
- Neuroleptically induced dystonia in Huntington's disease: a case report. Schott, K., Ried, S., Stevens, I., Dichgans, J. Eur. Neurol. (1989)
- Effects of tiapride on electroencephalograms and cognitive functions in the elderly. Patat, A., Alberini, H., Bonhomme, D., Soubrane, C., Allain, H., Gandon, J.M. International clinical psychopharmacology. (1999)
- Treatment of alcohol withdrawal syndrome with a combination of tiapride/carbamazepine : Results of a pooled analysis in 540 patients. Soyka, M., Schmidt, P., Franz, M., Barth, T., de Groot, M., Kienast, T., Reinert, T., Richter, C., Sander, G. European archives of psychiatry and clinical neuroscience. (2006)