Chemical Compound Review:
Tryptamin 2-(1H-indol-3-yl)ethanamine
Synonyms:
tryptamine, PubChem9450, CHEMBL6640, SureCN26725, AGN-PC-006Z67, ...
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- Stability of Lambdoid bacteriophage heads: antagonism between polyamines and tryptamine. Deeb, S.S., Moyle, E.A. J. Virol. (1982)
- Tryptamine induces phosphoinositide turnover and modulates adrenergic and muscarinic cholinergic receptor function in cultured cerebellar granule cells. Ishitani, R., Kimura, M., Takeichi, M., Chuang, D.M. J. Neurochem. (1994)
- High-performance liquid-chromatographic analysis for serotonin and tryptamine excreted in urine after oral loading with L-tryptophan. Tsuchiya, H., Hayashi, T., Tatsumi, M., Hoshino, Y., Ohtani, S., Takagi, N. Clin. Chem. (1989)
- Region-selective decreases in densities of [3H]tryptamine binding sites in autopsied brain tissue from cirrhotic patients with hepatic encephalopathy. Mousseau, D.D., Layrargues, G.P., Butterworth, R.F. J. Neurochem. (1994)
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- Tryptamine: a neuromodulator or neurotransmitter in mammalian brain? Jones, R.S. Prog. Neurobiol. (1982)
- Histological localization of messenger RNAs for rat acetyltransferases that acetylate serotonin and genotoxic arylamines. Debiec-Rychter, M., Land, S.J., King, C.M. Cancer Res. (1996)
- Expression of enzymatically active cloned strictosidine synthase from the higher plant Rauvolfia serpentina in Escherichia coli. Kutchan, T.M. FEBS Lett. (1989)
- Tryptamine-induced myoclonus in guinea-pigs pretreated with a monoamine oxidase inhibitor indicates pre- and post-synaptic actions of tryptamine upon central indoleamine systems. Luscombe, G., Jenner, P., Marsden, C.D. Neuropharmacology (1982)
- In vitro and in vivo characterization of the dopamine D4 receptor, serotonin 5-HT2A receptor and alpha-1 adrenoceptor antagonist (R)-(+)-2-amino-4-(4-fluorophenyl)-5-[1-[4-(4-fluorophenyl)-4-oxobutyl] pyrrolidin-3-yl]thiazole (NRA0045). Okuyama, S., Chaki, S., Yoshikawa, R., Suzuki, Y., Ogawa, S., Imagawa, Y., Kawashima, N., Ikeda, Y., Kumagai, T., Nakazato, A., Nagamine, M., Tomisawa, K. J. Pharmacol. Exp. Ther. (1997)
- F 11356, a novel 5-hydroxytryptamine (5-HT) derivative with potent, selective, and unique high intrinsic activity at 5-HT1B/1D receptors in models relevant to migraine. John, G.W., Pauwels, P.J., Perez, M., Halazy, S., Le Grand, B., Verscheure, Y., Valentin, J.P., Palmier, C., Wurch, T., Chopin, P., Marien, M., Kleven, M.S., Koek, W., Assie, M.B., Carilla-Durand, E., Tarayre, J.P., Colpaert, F.C. J. Pharmacol. Exp. Ther. (1999)
- Highly efficient Lewis acid-catalysed Pictet-Spengler reactions discovered by parallel screening. Srinivasan, N., Ganesan, A. Chem. Commun. (Camb.) (2003)
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- Complete amino acid analysis of proteins from a single hydrolysate. Simpson, R.J., Neuberger, M.R., Liu, T.Y. J. Biol. Chem. (1976)
- Arylamine N-methyltransferase. Methylation of the indole ring. Lyon, E.S., Jakoby, W.B. J. Biol. Chem. (1982)
- Targeting tryptophan decarboxylase to selected subcellular compartments of tobacco plants affects enzyme stability and in vivo function and leads to a lesion-mimic phenotype. Di Fiore, S., Li, Q., Leech, M.J., Schuster, F., Emans, N., Fischer, R., Schillberg, S. Plant Physiol. (2002)
- X-ray crystallographic studies of serotonin N-acetyltransferase catalysis and inhibition. Wolf, E., De Angelis, J., Khalil, E.M., Cole, P.A., Burley, S.K. J. Mol. Biol. (2002)
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- Central tryptamine turnover in depression, schizophrenia, and anorexia: measurement of indoleacetic acid in cerebrospinal fluid. Anderson, G.M., Gerner, R.H., Cohen, D.J., Fairbanks, L. Biol. Psychiatry (1984)
- Benzodiazepine receptor affinity and interaction of some N-(indol-3-ylglyoxylyl)amine derivatives. Bianucci, A.M., Da Settimo, A., Da Settimo, F., Primofiore, G., Martini, C., Giannaccini, G., Lucacchini, A. J. Med. Chem. (1992)
- Effect of intranigral administration of 6-hydroxydopamine and 5,7-dihydroxytryptamine on rat brain tryptamine. Juorio, A.V., Greenshaw, A.J., Nguyen, T.V. J. Neurochem. (1987)
- Tryptamine: a possible endogenous substrate for CYP2D6. Martínez, C., Agúndez, J.A., Gervasini, G., Martín, R., Benítez, J. Pharmacogenetics (1997)
- Ligands which effect human protein C activation by thrombin. Musci, G., Berliner, L.J. J. Biol. Chem. (1987)
- Amphetamine, 3,4-methylenedioxymethamphetamine, lysergic acid diethylamide, and metabolites of the catecholamine neurotransmitters are agonists of a rat trace amine receptor. Bunzow, J.R., Sonders, M.S., Arttamangkul, S., Harrison, L.M., Zhang, G., Quigley, D.I., Darland, T., Suchland, K.L., Pasumamula, S., Kennedy, J.L., Olson, S.B., Magenis, R.E., Amara, S.G., Grandy, D.K. Mol. Pharmacol. (2001)
- Interaction of tryptamine and ergoline compounds with threonine 196 in the ligand binding site of the 5-hydroxytryptamine6 receptor. Boess, F.G., Monsma, F.J., Meyer, V., Zwingelstein, C., Sleight, A.J. Mol. Pharmacol. (1997)
- Evidence that 5-methoxy-N, N-dimethyl tryptamine is a specific substrate for MAO-A in the rat: implications for the indoleamine dependent behavioural syndrome. Squires, R.F. J. Neurochem. (1975)
- Serotoninergic system in hamster skin. Slominski, A., Pisarchik, A., Semak, I., Sweatman, T., Szczesniewski, A., Wortsman, J. J. Invest. Dermatol. (2002)
- Interactions of tryptamine derivatives with serotonin transporter species variants implicate transmembrane domain I in substrate recognition. Adkins, E.M., Barker, E.L., Blakely, R.D. Mol. Pharmacol. (2001)
- Modulation of CYP1A2 enzyme activity by indoleamines: inhibition by serotonin and tryptamine. Agúndez, J.A., Gallardo, L., Martínez, C., Gervasini, G., Benítez, J. Pharmacogenetics (1998)
- Human indolethylamine N-methyltransferase: cDNA cloning and expression, gene cloning, and chromosomal localization. Thompson, M.A., Moon, E., Kim, U.J., Xu, J., Siciliano, M.J., Weinshilboum, R.M. Genomics (1999)
- Purification of endogenous modulators of monoamine oxidase from plasma. Giambalvo, C.T. Biochem. Pharmacol. (1984)
- Isolation, crystallization, and properties of indolyl-3-alkane alpha-hydroxylase. A novel tryptophan-metabolizing enzyme. Roberts, J., Rosenfeld, H.J. J. Biol. Chem. (1977)
- Determination of kinetic properties of serotonin-N-acetyltransferase in bovine pineal gland using HPLC with fluorimetric detection. Fajardo, N., Abreu, P., Alonso, R. J. Pineal Res. (1992)
- Effect of L-tryptophan on mouse brain 5-hydroxytryptamine: comparison of values obtained using a fluorimetric assay and a liquid Chromatographic assay with electrochemical detection. Marsden, C.A. J. Neurochem. (1981)