Chemical Compound Review:
Pevaryl 1-[2-[(4- chlorophenyl)methoxy]-2- (2,4...
Synonyms:
Econazol, Palavale, Ecostatin, econazole, Econazolum, ...
Hill,
McNulty,
Randall,
Nilius,
Prenen,
Vennekens,
Hoenderop,
Bindels,
Droogmans,
Hui,
Chan,
Barbadillo,
Lee,
Maibach,
Wester,
Schwarz,
Wissenbach,
Niemeyer,
Strauss,
Philipp,
Flockerzi,
Hoth,
Viana,
de Smedt,
Droogmans,
Nilius,
Xiao,
Huang,
Morgan,
Czeizel,
Kazy,
Vargha,
Ghelardi,
Tavanti,
Lupetti,
Celandroni,
Boldrini,
Campa,
Senesi,
Chen,
Bauer,
Kuchler,
Clark-Walker,
- Imidazole antifungals Miconazole and Econazole induce apoptosis in mouse lymphoma and human T cell leukemia cells: regulation by Bcl-2 and potential role of calcium. Sobecks, R., McCormick, T.S., Distelhorst, C.W. Cell Death Differ. (1996)
- Control of Candida albicans murine vaginitis by topical administration of polycarbophil-econazole complex. Ghelardi, E., Tavanti, A., Lupetti, A., Celandroni, F., Boldrini, E., Campa, M., Senesi, S. Antimicrob. Agents Chemother. (1998)
- Sulconazole. A review of its antimicrobial activity and therapeutic use in superficial dermatomycoses. Benfield, P., Clissold, S.P. Drugs (1988)
- A Parenteral Econazole Formulation Using a Novel Micelle-to-Liposome Transfer Method: In Vitro Characterization and Tumor Growth Delay in a Breast Cancer Xenograft Model. Cogswell, S., Berger, S., Waterhouse, D., Bally, M.B., Wasan, E.K. Pharm. Res. (2006)
- Purging of contaminating breast cancer cells from hematopoietic progenitor cell preparations using activation enhanced cell death. Zhang, Y., Crump, M., Berge, S.A. Breast Cancer Res. Treat. (2002)
- A population-based case-control teratological study of vaginal econazole treatment during pregnancy. Czeizel, A.E., Kazy, Z., Vargha, P. Eur. J. Obstet. Gynecol. Reprod. Biol. (2003)
- Isolation of a full-length cDNA insert encoding human aromatase system cytochrome P-450 and its expression in nonsteroidogenic cells. Corbin, C.J., Graham-Lorence, S., McPhaul, M., Mason, J.I., Mendelson, C.R., Simpson, E.R. Proc. Natl. Acad. Sci. U.S.A. (1988)
- Cytochrome P450 may regulate plasma membrane Ca2+ permeability according to the filling state of the intracellular Ca2+ stores. Alvarez, J., Montero, M., Garcia-Sancho, J. FASEB J. (1992)
- Increased calcium influx and ribosomal content correlate with resistance to endoplasmic reticulum stress-induced cell death in mutant leukemia cell lines. Zhang, Y., Berger, S.A. J. Biol. Chem. (2004)
- Intracellular mediators of granulysin-induced cell death. Okada, S., Li, Q., Whitin, J.C., Clayberger, C., Krensky, A.M. J. Immunol. (2003)
- C-mitosis and numerical chromosome aberration analyses in human lymphocytes: 10 known or suspected spindle poisons. Sbrana, I., Di Sibio, A., Lomi, A., Scarcelli, V. Mutat. Res. (1993)
- On the mechanism of action of econazole, the capacitative calcium inflow blocker. Gamberucci, A., Fulceri, R., Benedetti, A., Bygrave, F.L. Biochem. Biophys. Res. Commun. (1998)
- Naftifine cream 1% versus econazole cream 1% in the treatment of tinea cruris and tinea corporis. Millikan, L.E., Galen, W.K., Gewirtzman, G.B., Horwitz, S.N., Landow, R.K., Nesbitt, L.T., Roth, H.L., Sefton, J., Day, R.M. J. Am. Acad. Dermatol. (1988)
- Three-day therapy of vaginal candidiasis with clotrimazole vaginal tablets and econazole ovules: a multicenter comparative study. Stettendorf, S., Benijts, G., Vignali, M., Kreysing, W. Chemotherapy. (1982)
- Treatment of candidal vaginitis. A prospective randomized investigator-blind multicenter study comparing topically applied econazole with oral fluconazole. Osser, S., Haglund, A., Weström, L. Acta obstetricia et gynecologica Scandinavica. (1991)
- Stimulation of HIV expression by intracellular calcium pump inhibition. Papp, B., Byrn, R.A. J. Biol. Chem. (1995)
- Extracellular site for econazole-mediated block of Ca2+ release-activated Ca2+ current (Icrac) in T lymphocytes. Christian, E.P., Spence, K.T., Togo, J.A., Dargis, P.G., Warawa, E. Br. J. Pharmacol. (1996)
- TRPV6 potentiates calcium-dependent cell proliferation. Schwarz, E.C., Wissenbach, U., Niemeyer, B.A., Strauss, B., Philipp, S.E., Flockerzi, V., Hoth, M. Cell Calcium (2006)
- Econazole, a blocker of Ca2+ influx, selectively suppresses LTP of EPSPs in hippocampal slices. Forghani, R., Krnjević, K. Neurosci. Lett. (1995)
- Inhibitory effect of purines in meiotic maturation of denuded mouse oocytes. Shim, C., Lee, D.K., Lee, C.C., Cho, W.K., Kim, K. Mol. Reprod. Dev. (1992)
- Econazole inhibits thapsigargin-induced platelet calcium influx by mechanisms other than cytochrome P-450 inhibition. Vostal, J.G., Fratantoni, J.C. Biochem. J. (1993)
- Cytochrome P450: a novel system modulating Ca2+ channels and contraction in mammalian heart cells. Xiao, Y.F., Huang, L., Morgan, J.P. J. Physiol. (Lond.) (1998)
- Effects of staurosporine on the capacitative regulation of the state of the Ca2+ reserves in activated Jurkat T lymphocytes. Ahnadi, C.E., Payet, M.D., Dupuis, G. Cell Calcium (1996)
- Sensitivity of myeloid leukemia cells to calcium influx blockade: application to bone marrow purging. Soboloff, J., Zhang, Y., Minden, M., Berger, S.A. Exp. Hematol. (2002)
- Positive and negative control of multidrug resistance by the Sit4 protein phosphatase in Kluyveromyces lactis. Chen, X.J., Bauer, B.E., Kuchler, K., Clark-Walker, G.D. J. Biol. Chem. (2000)
- Transcriptional regulation of rat microsomal epoxide hydrolase gene by imidazole antimycotic agents. Kim, S.G. Mol. Pharmacol. (1992)
- Cloning and characterization of CYP51 from Mycobacterium avium. Pietila, M.P., Vohra, P.K., Sanyal, B., Wengenack, N.L., Raghavakaimal, S., Thomas, C.F. Am. J. Respir. Cell Mol. Biol. (2006)
- Use of decimal assay for additivity to demonstrate synergy in pair combinations of econazole, nikkomycin Z, and ibuprofen against Candida albicans in vitro. Tariq, V.N., Scott, E.M., McCain, N.E. Antimicrob. Agents Chemother. (1995)
- In-vitro antifungal activity of sertaconazole, bifonazole, ketoconazole, and miconazole against yeasts of the Candida genus. Carrilo-Muñoz, A.J., Tur, C., Torres, J. J. Antimicrob. Chemother. (1996)
- Thapsigargin-stimulated MAP kinase phosphorylation via CRAC channels and PLD activation: inhibitory action of docosahexaenoic acid. Denys, A., Aires, V., Hichami, A., Khan, N.A. FEBS Lett. (2004)
- Pharmacological modulation of monovalent cation currents through the epithelial Ca2+ channel ECaC1. Nilius, B., Prenen, J., Vennekens, R., Hoenderop, J.G., Bindels, R.J., Droogmans, G. Br. J. Pharmacol. (2001)
- Pituitary adenylate cyclase-activating polypeptide induces a sustained increase in intracellular free Ca(2+) concentration and catechol amine release by activating Ca(2+) influx via receptor-stimulated Ca(2+) entry, independent of store-operated Ca(2+) channels, and voltage-dependent Ca(2+) channels in bovine adrenal medullary chromaffin cells. Morita, K., Sakakibara, A., Kitayama, S., Kumagai, K., Tanne, K., Dohi, T. J. Pharmacol. Exp. Ther. (2002)
- Calcium signalling through nucleotide receptor P2Y2 in cultured human vascular endothelium. Viana, F., de Smedt, H., Droogmans, G., Nilius, B. Cell Calcium (1998)
- Inhibition of TRPM2 channels by the antifungal agents clotrimazole and econazole. Hill, K., McNulty, S., Randall, A.D. Naunyn Schmiedebergs Arch. Pharmacol. (2004)
- Calcium influx evoked by Ca2+ store depletion in human platelets is more susceptible to cytochrome P-450 inhibitors than receptor-mediated calcium entry. Sargeant, P., Clarkson, W.D., Sage, S.O., Heemskerk, J.W. Cell Calcium (1992)
- Enhanced econazole penetration into human nail by 2-n-nonyl-1,3-dioxolane. Hui, X., Chan, T.C., Barbadillo, S., Lee, C., Maibach, H.I., Wester, R.C. Journal of pharmaceutical sciences. (2003)
- Efficacy of econazole ('Gyno-Pevaryl' 150) in vaginal candidosis during pregnancy. Goormans, E., Beek, J.M., Declercq, J.A., Loendersloot, E.W., Roelofs, H.J., van Zanten, A. Current medical research and opinion. (1985)