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Chemical Compound Review

Regitine     3-[4,5-dihydro-1H-imidazol-2- ylmethyl-(4...

Synonyms: Regitina, Regitipe, Rogitine, Dibasin, Regitin, ...
 
 
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Disease relevance of phentolamine

 

Psychiatry related information on phentolamine

 

High impact information on phentolamine

 

Chemical compound and disease context of phentolamine

 

Biological context of phentolamine

 

Anatomical context of phentolamine

 

Associations of phentolamine with other chemical compounds

 

Gene context of phentolamine

  • Neither tetrodotoxin (TTX) nor phentolamine affected responses to either NPY or PYY on the jejunum [36].
  • While the pressor response to ET-1 was significantly inhibited after i.v. injection of phentolamine, the bradycardia was blocked by pentolinium [37].
  • Contractions to SRIF were not antagonised by the putative SRIF receptor blocker cyclo(7-aminoheptanoyl-Phe-D Trp-Lys-Thr[Bzl]) (CPP), phentolamine, or indomethacin [38].
  • GHRH alone and combined with i.v. infusion of phentolamine (PHEN), alpha 1/alpha 2-antagonist, (0.5 mg/min from -60 to +30 min); 5 [39].
  • However, in contrast to RG20, [3H] rauwolscine exhibits a KD of 2 nM for the C-10 receptor, and the potency order for competing ligands is rauwolscine greater than or equal to yohimbine greater than idazoxan greater than phentolamine greater than prazosin [40].
 

Analytical, diagnostic and therapeutic context of phentolamine

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