Chemical Compound Review:
fentanyl N-(1-phenethyl-4-piperidyl)- N-phenyl...
Synonyms:
Fentanil, Matrifen, Pentanyl, Sentonil, Duragesic, ...
- Transdermal fentanyl for postoperative pain management. A double-blind placebo study. Caplan, R.A., Ready, L.B., Oden, R.V., Matsen, F.A., Nessly, M.L., Olsson, G.L. JAMA (1989)
- Hypotension with midazolam and fentanyl in the newborn. Burtin, P., Daoud, P., Jacqz-Aigrain, E., Mussat, P., Moriette, G. Lancet (1991)
- Carbon dioxide retention and oxygen desaturation during gastrointestinal endoscopy. Freeman, M.L., Hennessy, J.T., Cass, O.W., Pheley, A.M. Gastroenterology (1993)
- Randomised trial of fentanyl anaesthesia in preterm babies undergoing surgery: effects on the stress response. Anand, K.J., Sippell, W.G., Aynsley-Green, A. Lancet (1987)
- Fedotozine reverses ileus induced by surgery or peritonitis: action at peripheral kappa-opioid receptors. Rivière, P.J., Pascaud, X., Chevalier, E., Le Gallou, B., Junien, J.L. Gastroenterology (1993)
- Trends in medical use and abuse of opioid analgesics. Joranson, D.E., Ryan, K.M., Gilson, A.M., Dahl, J.L. JAMA (2000)
- Severe deficit in brain reward function associated with fentanyl withdrawal in rats. Bruijnzeel, A.W., Lewis, B., Bajpai, L.K., Morey, T.E., Dennis, D.M., Gold, M. Biol. Psychiatry (2006)
- Relief of persistent postamputation stump and phantom limb pain with intrathecal fentanyl. Jacobson, L., Chabal, C., Brody, M.C. Pain (1989)
- Postoperative sleep disturbance: influences of opioids and pain in humans. Cronin, A.J., Keifer, J.C., Davies, M.F., King, T.S., Bixler, E.O. Sleep. (2001)
- Profiles of opioid analgesia in humans after intravenous bolus administration: alfentanil, fentanyl and morphine compared on experimental pain. Chapman, C.R., Hill, H.F., Saeger, L., Gavrin, J. Pain (1990)
- Preemptive epidural analgesia and recovery from radical prostatectomy: a randomized controlled trial. Gottschalk, A., Smith, D.S., Jobes, D.R., Kennedy, S.K., Lally, S.E., Noble, V.E., Grugan, K.F., Seifert, H.A., Cheung, A., Malkowicz, S.B., Gutsche, B.B., Wein, A.J. JAMA (1998)
- Nosocomial Pseudomonas pickettii bacteremias traced to narcotic tampering. A case for selective drug screening of health care personnel. Maki, D.G., Klein, B.S., McCormick, R.D., Alvarado, C.J., Zilz, M.A., Stolz, S.M., Hassemer, C.A., Gould, J., Liegel, A.R. JAMA (1991)
- Nociceptin/orphanin FQ exacerbates excitotoxic white-matter lesions in the murine neonatal brain. Laudenbach, V., Calo, G., Guerrini, R., Lamboley, G., Benoist, J.F., Evrard, P., Gressens, P. J. Clin. Invest. (2001)
- Randomised double-blind active-placebo-controlled crossover trial of intravenous fentanyl in neuropathic pain. Dellemijn, P.L., Vanneste, J.A. Lancet (1997)
- Progressive hypoxemia limits left ventricular oxygen consumption and contractility. Walley, K.R., Becker, C.J., Hogan, R.A., Teplinsky, K., Wood, L.D. Circ. Res. (1988)
- Reduction of cerebrospinal fluid pressure by hypocapnia: changes in cerebral blood volume, cerebrospinal fluid volume and brain tissue water and electrolytes. II. Effects of anesthetics. Artru, A.A. J. Cereb. Blood Flow Metab. (1988)
- Anesthetic modulation of cerebral hemodynamic and evoked responses to transient middle cerebral artery occlusion in cats. Helfaer, M.A., Kirsch, J.R., Traystman, R.J. Stroke (1990)
- The role of neuronal nitric oxide synthase in regulation of cerebral blood flow in normocapnia and hypercapnia in rats. Wang, Q., Pelligrino, D.A., Baughman, V.L., Koenig, H.M., Albrecht, R.F. J. Cereb. Blood Flow Metab. (1995)
- Safety and efficacy of xenon in routine use as an inhalational anaesthetic. Lachmann, B., Armbruster, S., Schairer, W., Landstra, M., Trouwborst, A., Van Daal, G.J., Kusuma, A., Erdmann, W. Lancet (1990)
- Acute respiratory acidosis decreases left ventricular contractility but increases cardiac output in dogs. Walley, K.R., Lewis, T.H., Wood, L.D. Circ. Res. (1990)
- In vivo studies of opiate receptors. Frost, J.J., Dannals, R.F., Duelfer, T., Burns, H.D., Ravert, H.T., Langström, B., Balasubramanian, V., Wagner, H.N. Ann. Neurol. (1984)
- Mu Opioid Receptor Activation of ERK1/2 Is GRK3 and Arrestin Dependent in Striatal Neurons. Macey, T.A., Lowe, J.D., Chavkin, C. J. Biol. Chem. (2006)
- Randomised comparison of combined spinal-epidural and standard epidural analgesia in labour. Collis, R.E., Davies, D.W., Aveling, W. Lancet (1995)
- Unilateral analgesia following injection of fentanyl into the lumbosacral plexus. Smith, B., Pinnock, C., Fischer, B., Trotter, T., Scott, P. Lancet (1987)
- beta-Arrestin2, interacting with phosphodiesterase 4, regulates synaptic release probability and presynaptic inhibition by opioids. Bradaïa, A., Berton, F., Ferrari, S., Lüscher, C. Proc. Natl. Acad. Sci. U.S.A. (2005)
- Diastolic viscous properties of the intact canine left ventricle. Nikolic, S.D., Tamura, K., Tamura, T., Dahm, M., Frater, R.W., Yellin, E.L. Circ. Res. (1990)
- Passive properties of canine left ventricle: diastolic stiffness and restoring forces. Nikolić, S., Yellin, E.L., Tamura, K., Vetter, H., Tamura, T., Meisner, J.S., Frater, R.W. Circ. Res. (1988)
- Rapid switching between transdermal fentanyl and methadone in cancer patients. Mercadante, S., Ferrera, P., Villari, P., Casuccio, A. J. Clin. Oncol. (2005)
- Neuroleptanalgesia in upper alimentary endoscopy. Le Brun, H.I. Gut (1976)
- Elective bedside surgery in critically injured patients is safe and cost-effective. Van Natta, T.L., Morris, J.A., Eddy, V.A., Nunn, C.R., Rutherford, E.J., Neuzil, D., Jenkins, J.M., Bass, J.G. Ann. Surg. (1998)
- Pharmacokinetics of midazolam, propofol, and fentanyl transfer to human breast milk. Nitsun, M., Szokol, J.W., Saleh, H.J., Murphy, G.S., Vender, J.S., Luong, L., Raikoff, K., Avram, M.J. Clin. Pharmacol. Ther. (2006)
- Pharmacokinetic-pharmacodynamic modeling in drug development: application to the investigational opioid trefentanil. Lemmens, H.J., Dyck, J.B., Shafer, S.L., Stanski, D.R. Clin. Pharmacol. Ther. (1994)
- Agonist induced homologous desensitization of mu-opioid receptors mediated by G protein-coupled receptor kinases is dependent on agonist efficacy. Kovoor, A., Celver, J.P., Wu, A., Chavkin, C. Mol. Pharmacol. (1998)
- Possible involvement of multiple cytochrome P450S in fentanyl and sufentanil metabolism as opposed to alfentanil. Guitton, J., Buronfosse, T., Désage, M., Lepape, A., Brazier, J.L., Beaune, P. Biochem. Pharmacol. (1997)
- Influence of the menstrual cycle on neuroendocrine and behavioral responses to an opiate agonist in humans: preliminary results. Hoehe, M. Psychoneuroendocrinology (1988)
- Remifentanil directly activates human N-methyl-D-aspartate receptors expressed in Xenopus laevis oocytes. Hahnenkamp, K., Nollet, J., Van Aken, H.K., Buerkle, H., Halene, T., Schauerte, S., Hahnenkamp, A., Hollmann, M.W., Strümper, D., Durieux, M.E., Hoenemann, C.W. Anesthesiology (2004)
- Simultaneous assessment of drug interactions with low- and high-extraction opioids: application to parecoxib effects on the pharmacokinetics and pharmacodynamics of fentanyl and alfentanil. Ibrahim, A.E., Feldman, J., Karim, A., Kharasch, E.D. Anesthesiology (2003)
- Narcotic analgesia: fentanyl reduces the intensity but not the unpleasantness of painful tooth pulp sensations. Gracely, R.H., Dubner, R., McGrath, P.A. Science (1979)
- Valvular-ventricular interaction: importance of the mitral apparatus in canine left ventricular systolic performance. Hansen, D.E., Cahill, P.D., DeCampli, W.M., Harrison, D.C., Derby, G.C., Mitchell, R.S., Miller, D.C. Circulation (1986)
- Opiate drugs and delta-receptor-mediated myocardial protection. Benedict, P.E., Benedict, M.B., Su, T.P., Bolling, S.F. Circulation (1999)